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N-[(2R,3R)-1'-[(3,7-dimethyl-1H-indol-2-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
3-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrazine-2-carbonitrile
3-methanesulfonyl-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[4-(trifluoromethoxy)benzenesulfonyl]piperidine
(4aR,8aS)-1-(2,2-diphenylethyl)-6-[2-(3,4,5-trimethoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-[(dimethylamino)methyl]-N,N-bis(1,3-oxazol-4-ylmethyl)benzamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1-cyclopentylpiperidine-3-carboxamide
3-(5-pentyl-1,3,4-thiadiazol-2-yl)-1-(thiolan-3-yl)urea
5-(3-acetylphenoxymethyl)-N-(1-benzylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
4-(2-oxopyrrolidin-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butanamide
1-(3-methoxyphenyl)-4-(2-phenoxypropanoyl)piperazin-2-one
1-[2-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-methylazepane-2-carboxamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(6-hydroxy-6-methylheptan-2-yl)piperidine-4-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,7S)-3-(2-phenoxyethyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxylate
1-(furan-2-ylmethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpiperidine-3-carboxamide
2-ethyl-N-[(4-fluorophenyl)methyl]-4-methyl-N-(pyridin-4-ylmethyl)-1,3-oxazole-5-carboxamide
1-(cyclopropylmethyl)-4-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-(propan-2-yl)-1,4-diazepane
5-(3-chloro-4-fluorophenyl)pyrimidin-2-amine
(3S,4R)-1-(3-fluoropyridin-4-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
1-[4-phenyl-1-(thiophen-3-ylmethyl)piperidin-4-yl]ethan-1-one
6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
3-(2-ethylphenoxy)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}azetidine
5-(2-methylphenyl)-4-[1-(naphthalene-2-carbonyl)piperidin-3-yl]-2-(pyridin-4-yl)pyrimidine
3-{1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]azetidin-3-yl}pyridine
(4aS,7aR)-1-(5-hydroxypyrazine-2-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(2-chlorophenyl)methyl]-5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-(3-fluorophenyl)-6-[(4-methylphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
N-(3-hydroxyadamantan-1-yl)-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
N-(1-{4-[4-(quinazolin-4-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)oxolane-3-carboxamide
4-(1,3-benzothiazol-2-yl)-2-({[2-(4-fluorophenyl)ethyl]amino}methyl)phenol
{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-(1H-imidazol-1-ylmethyl)-1-(5-methyl-1-benzofuran-2-carbonyl)piperidin-4-ol
ethyl 1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-butyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1,3-benzoxazole
3-(1-benzothiophen-3-yl)-1-methyl-6-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-methyl-1H-1,3-benzodiazole-4-carboxamide
1-ethyl-6-oxo-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
3-[5-(2,4-dichlorophenyl)-4-phenyl-1H-imidazol-1-yl]propane-1,2-diol
4-[(5-acetyl-4-methylpyrimidin-2-yl)amino]-1-(3-chlorophenyl)pyrrolidin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
3-(4-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid