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3-methoxy-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
2-chloro-5-acetamido-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
N-[4-fluoro-3-(methylcarbamoyl)phenyl]-3-(methoxymethyl)pyrrolidine-1-carboxamide
5-fluoro-3-{[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1H-indole
N,N-dimethyl-1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carboxamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-4-(3-hydroxy-3-methylbutyl)benzamide
N-butyl-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]benzamide
methyl 1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxylate
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
(3aR,6aR)-2-methyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
N-ethyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pentan-3-yl)acetamide
5-(hydroxymethyl)-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-methoxy-2-(thiophen-2-yl)ethyl]amine
5,6-dimethyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
4-(2-fluorophenoxy)-1-(1,3-thiazol-4-ylmethyl)piperidine
2-{3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}pyrrolidine-1-carboxamide
2-[1-(1-methylpiperidin-4-yl)-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[(3-acetylphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(3,4,5-trimethoxyphenyl)acetamide
(2E)-1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
1-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
7-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxypropanamide
(1S,5R)-6-(3,4-dimethylbenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-(2,4-dichlorophenoxy)-1-[3-(propoxymethyl)pyrrolidin-1-yl]ethan-1-one
1-[2-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)ethyl]azepan-2-one
2-[3-(4-ethylphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-(butan-2-yl)-3-(3,4-difluorophenyl)-N-(pyridin-4-ylmethyl)propanamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(2-methylpropyl)imidazo[1,2-a]pyrimidine-3-carboxamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-(morpholin-4-yl)benzamide
1-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}piperidin-3-ol
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-methoxypyridine
[2-(2-fluorophenyl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-methyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{1-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N,2-dimethylfuran-3-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(pyrazin-2-yl)propanamide
1-{7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-(4-methoxyphenyl)-6,6-dimethyl-4-[3-(methylsulfanyl)propanoyl]piperazin-2-one
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-[(2R,3R)-1'-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
3-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-1-ol
(9aR)-N-(3-fluorophenyl)-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-ethyl-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]pyridine-3-carboxamide
methyl 9-(benzyloxy)-3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine