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1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
methyl 4-[4-({[(1-ethyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
(4aS,8aR)-6-(dimethyl-1,3-oxazole-4-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}propanamide
3-{5-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
2-[4-(1H-pyrazol-1-yl)phenyl]-4-(pyrrolidine-1-carbonyl)pyridine
2-{1-[1-(3,5,5-trimethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methyl-3-[methyl(propan-2-yl)amino]propan-1-one
8-(3-ethyl-1H-pyrazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-N'-ethyl-N'-(pyridin-4-ylmethyl)butanediamide
(2E)-3-phenyl-1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
2-{2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(3S,4S)-1-(azepane-1-sulfonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-methoxyphenyl)piperidine
(3aS,6aS)-2-(ethanesulfonyl)-5-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-methoxyphenyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-4-oxobutanamide
N-(cyclopropylmethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}[(2-fluorophenyl)methyl]amine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxymethyl]piperidin-1-yl}ethan-1-one
3-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
(2S,4R)-N-[2-(dimethylamino)ethyl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
N-[(3S,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
4-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-(morpholin-4-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}benzamide
2-(2,4,5-trifluorobenzenesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(4-hydroxyphenyl)methyl]-3,5-dimethyladamantane-1-carboxamide
3-[2-(dimethylamino)ethyl]-1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrazol-5-yl)urea
methyl N-{2-[2-methyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]-2-oxoethyl}carbamate
9-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-fluorophenyl)methyl]-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-benzyl-3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(2-hydroxyethyl)propanamide
methyl 3-(4-methoxybenzamido)-1-methyl-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(furan-3-ylmethyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-methoxyethyl)-2,7-dimethyl-N-(1-methylpiperidin-4-yl)quinoline-4-carboxamide
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-2,3-dihydro-1H-isoindole
4-(2-fluorophenoxy)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-[3-(2-cyclopropyl-1H-imidazol-1-yl)propyl]-4,5-dimethyl-1H-1,3-benzodiazole
1-(2-methyl-4-{[3-(oxolan-3-yl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-N-[(2,4,6-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(pyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
6-methoxy-N-[(5-methoxy-1H-indol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(thiophene-2-carbonyl)piperidine