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7-(2-methylphenyl)-4-[2-(morpholin-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[(1R,5S,6R)-3-(furan-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}(methyl)[3-(1-methyl-1H-pyrazol-4-yl)propyl]amine
8-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
5-[3-(azocan-1-yl)-3-oxopropyl]-5-[(4-fluorophenyl)methyl]pyrrolidin-2-one
N-({7-[2-(2,3,6-trifluorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)cyclopropanecarboxamide
N-methyl-N-(1-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
1-(cyclopropylmethyl)-5-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{3-[3-(3,4-dimethoxyphenyl)phenyl]-1H-pyrazol-1-yl}acetamide
1-(2-phenylethyl)-3-(propan-2-yl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
7-(7-chloro-4-methylquinolin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-indole-6-carboxamide
6-methoxy-2-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N,2,2,6,6-pentamethyl-N-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-amine
2-({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-5-methoxy-N-methyl-1H-indole-2-carboxamide
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
1-[(2-methoxyphenyl)methyl]-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine-3-carboxylate
4-[4-(4-methoxybenzoyl)piperazin-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1-cyclobutanecarbonylpiperidine
2-({2-amino-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-(1-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-[5-(3-ethyl-5-methyl-1,2-oxazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
4-(3-methylbut-2-en-1-yl)-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
1-benzyl-4-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-6-ol
methyl (2R)-2-[(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propanoate
1-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]azepan-4-amine
ethyl 2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-1,3-oxazole-4-carboxylate
N-(2-fluoroethyl)-3-{[(1R,2S)-2-phenylcyclopropyl]sulfamoyl}benzamide
3-(2,1,3-benzothiadiazol-5-ylmethyl)-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
8-(5-acetylthiophene-2-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(1,3-benzoxazol-2-yl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[2-(adamantan-1-yl)propan-2-yl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
ethyl 4-[(4-{[1-(thiophene-2-sulfonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
N3-[2-(cyclohex-1-en-1-yl)ethyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-4-(4-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
3-(1H-1,3-benzodiazol-2-yl)-N-[(4-hydroxyazepan-4-yl)methyl]propanamide
methyl 5-(3-methanesulfonamidopropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-{5-[(1S)-1-amino-2-(4-hydroxyphenyl)ethyl]-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-3-yl}acetamide
4-{1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-methylpropan-2-yl}morpholine
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2,7,8-trimethylquinoline-4-carboxamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-({[(2,6-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one