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[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](2-methoxyethyl)methylamine
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl}propanamide
N-tert-butyl-5-chloro-2-[(1-methylpiperidin-4-yl)oxy]benzamide
3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1-methyl-1,4-dihydroquinolin-4-one
2-{[2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-4-methoxyphenol
(2E)-3-(3,4-difluorophenyl)-1-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}prop-2-en-1-one
1-cyclohexyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidine-4-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(3-methylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
1-({5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]furan-2-yl}methyl)-1H-pyrazole
methyl 2-[(2-cyclohexyl-1,3-benzoxazol-6-yl)formamido]-4-(methylsulfanyl)butanoate
3-(1-methyl-1H-pyrrol-2-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-methyl-2-(2-methylpropanamido)benzamide
2-(dimethyl-1,3-thiazol-4-yl)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]acetamide
2-{4-[2-(methylsulfanyl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
methyl 1-methoxy-2-oxo-8-(3-phenyl-1,2-oxazole-5-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(3-{1-[(3-methoxyphenyl)methyl]-1H-pyrazol-3-yl}phenyl)-3-methylpyrazine
(1S,2R)-N1-(isoquinolin-5-ylmethyl)-N1-methyl-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
3-methyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
N-[(3R,4S)-1-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(3-{[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]methyl}pyridin-2-yl)piperidin-3-ol
(2E)-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
(2E)-3-(4-fluorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-butyl-N-methyl-3-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
ethyl 4-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
[1-(3-methylthiophene-2-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
N-(5-methoxy-2-methylphenyl)-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
1-cyclopropyl-3-(2-methylphenyl)-3-{2-oxo-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]ethyl}pyrrolidine-2,5-dione
7-(cyclohex-3-en-1-ylmethyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-[2-methyl-2-(piperidin-1-yl)propyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3S,5S,9S)-5-{[(4-methoxyphenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(pyrimidin-2-yl)piperazin-2-yl}ethan-1-ol
2-[(3,4-dimethoxyphenyl)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-(1-{2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(2,6-dimethoxypyridin-3-yl)urea
(2S,4S)-N,N-diethyl-4-(3-hydroxypropanamido)-1-(5-methylpyrazine-2-carbonyl)pyrrolidine-2-carboxamide
1-{[4-(methylsulfanyl)phenyl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]quinoxaline-5-carboxamide
5-[1-(4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-1,2,3-triazol-1-yl)ethyl]-1,3,4-thiadiazol-2-amine
(4aS,8aR)-1-(carboxymethyl)-6-[(2-methylphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[2-(dimethylamino)ethyl]-1-(6-fluoropyridin-3-yl)-3-[(5-methylthiophen-2-yl)methyl]urea
{4-[1-(9H-purin-6-yl)piperidin-4-yl]-1,4-oxazepan-6-yl}methanol
1-(2-methylphenyl)-4-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)piperazin-2-one
N-methyl-4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methylphenol
3-butyl-4-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-methylpiperazin-2-one
4-[4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]benzoic acid