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5-(4-methylpiperidine-1-carbonyl)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-(azepan-1-yl)-3-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-2-ol
4-{3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N-{2-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(thiophene-3-carbonyl)piperidine-4-carboxamide
1-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetyl]piperidine-4-carbonitrile
6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidine-2,4-diamine
1-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-phenylethane-1,2-dione
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
4-ethyl-1-[(1-methylpyrrolidin-3-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-methyl-1H-imidazol-5-yl)-4-(naphthalen-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-4-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1,3-oxazole-5-carboxamide
ethyl 1-benzyl-5-(4-hydroxybutan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{2-[2-(2,2-diphenylethyl)morpholin-4-yl]ethyl}dimethylamine
5-cyclopropyl-3-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(2-methoxyethyl)-9-[3-(1H-pyrazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-4-(methylsulfanyl)butan-1-one
3-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-(2-methoxyethyl)-N-methyl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]urea
5-[(3-fluorophenyl)methyl]-5-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
5-{[(2,6-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-hydroxy-4-methylbenzamide
(2S)-1-acetyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
(2R,3R,6R)-5-(ethanesulfonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{4-methyl-6-[3-(morpholin-4-ylmethyl)phenyl]pyrimidin-2-yl}phenol
2-{[(1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N-(3,4-difluorophenyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-fluorophenyl)acetamide
2-amino-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-6-(2-methylpropyl)pyrimidine-4-carboxamide
N-{[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
4-(hydroxymethyl)-1-[8-(trifluoromethyl)quinolin-4-yl]piperidin-4-ol
methyl 3-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidine-1-carbonyl)benzoate
1-(1,3-thiazol-2-ylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-{[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-[(2S,5R)-2,5-dimethylpiperazin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
5-(hydroxymethyl)-2-methyl-4-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-3-ol
2-(2,5-dimethoxyphenyl)-N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2,4-dichloro-3-{[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]methyl}phenol
1-cyclobutanecarbonyl-3-(2-fluorophenoxymethyl)piperidine
4-(4-{[2-(2-chlorophenyl)ethyl]amino}piperidin-1-yl)-N-cyclopentylbenzamide
N-{[3-(cyclopentyloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-4-(trifluoromethyl)benzamide
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
N-[2-(1H-pyrazol-1-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[(1-phenylcyclohexyl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-3-(2-hydroxyethyl)piperazin-2-one
N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3-(thiophen-2-yl)propanamide