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N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-[3-(pyridin-4-yl)propyl]acetamide
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(pyrrolidin-1-yl)acetamide
1-{4-[2-(3-phenylpropyl)morpholine-4-carbonyl]phenyl}ethan-1-one
5-ethyl-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2-oxazole-3-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl}methanol
2-[(3-chlorophenyl)methyl]-N-methyl-N-[3-(pyrrolidin-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
(4aR,7aS)-4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-propyl-5-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
[(3R,4R)-1-[(3-chloro-4-fluorophenyl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-[(5-chlorofuran-2-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
(2S,4S)-4-amino-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidine-2-carboxylic acid
1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
2-(3-chloro-4-fluorophenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
4-[(dipropylamino)methyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}benzamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(4-methoxyphenyl)-4-oxobutanamide
N-{3-methyl-1-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}furan-2-carboxamide
1-(cyclopropylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazin-2-yl}ethan-1-ol
6-[(diethylamino)methyl]-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazin-2-one
3-(3,4-difluorophenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-[2-(dimethylamino)ethyl]-1-[1-(2-fluorobenzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-[4-({4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-methyl-5-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}pyrimidin-2-amine
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
2-cyclopropyl-6-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
4-(3-methoxy-2-methylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(2-oxopyrrolidin-1-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}butanamide
(1R,5S)-6-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
1-{3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}-1H-1,2,3,4-tetrazole
5-{[(3-fluoro-4-methylphenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
ethyl 5-(1-benzofuran-2-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-methoxy-N-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
3-[(methylsulfanyl)methyl]-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazole
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-4-phenylbutan-1-one
1,2-dimethyl-5-[3-methyl-1-(3-methylbutyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
N-({1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
N,N-bis(propan-2-yl)-2-{thieno[2,3-d]pyrimidin-4-yl}benzamide
1-(3-methoxyphenyl)-4-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-2-one
N,N-dimethyl-4-{3-[1-(pyrrolidin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}benzamide
13-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
2-methyl-8-[(5-propylfuran-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione