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(2S,4R)-4-amino-N-ethyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidine-2-carboxamide
({1-[2-(2-fluorophenoxy)ethyl]-1H-indol-3-yl}methyl)(methyl)(1H-pyrazol-5-ylmethyl)amine
5-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
3-({7-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-(2,3-dihydro-1-benzofuran-7-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-ethyl-9-(3-methyl-1,2-oxazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-[1-benzyl-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-4,4,4-trifluorobutanamide
2-methyl-5-(3-methylphenyl)-4-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-3-yl]pyrimidine
1-(butan-2-yl)-N3-(2,3-dihydro-1H-inden-2-yl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})[1-(pyridin-3-yl)ethyl]amine
2-cyclopropyl-5-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyrimidine
1-(cyclohexylmethyl)-N-(oxolan-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-{2-methyl-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(carbamoylmethyl)-N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-4-carboxamide
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-[(2R,3R)-1'-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
3-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-1-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-methylurea
1-[(4-methoxyphenyl)methyl]-4-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-(cyclobutylmethyl)-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
9-[2-(2-chlorophenyl)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(azepan-1-yl)-3-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-{4-[5-(1H-1,3-benzodiazol-2-yl)furan-2-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
2-[4-(3-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-phenoxypropan-2-ol
1-(1-methyl-1H-pyrazole-5-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-(2,2-dimethyloxan-4-yl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
{1-[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperidin-4-yl}methanol
4-[methyl(oxan-2-ylmethyl)sulfamoyl]-N-(prop-2-en-1-yl)benzamide
N-methyl-3-{N-methyl-1-[3-(1H-pyrazol-4-yl)phenyl]formamido}propanamide
N-({7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
4-methyl-2-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-7-(methylsulfanyl)quinoline
8-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-{2-[cyclohexyl(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[1-(4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}phenyl)-1H-pyrazol-4-yl]-2,4-dimethylbenzamide
5-(3,4-difluorophenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-phenylethyl)urea
4-ethyl-N,N-dimethyl-6-(3,4,5-trimethoxyphenyl)pyrimidin-2-amine
N-[(2,3-difluoro-4-methylphenyl)methyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(ethanesulfonyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
1-{4-[(2-methoxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
7-[3-(furan-2-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
1-cyclopropyl-6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
5-{2-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
N-{4-[2-amino-3-cyano-6-(4-hydroxy-2-methylphenyl)pyridin-4-yl]phenyl}acetamide
7-fluoro-2-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione