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3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]propan-1-one
3-{[4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
N-[3-(1H-imidazol-1-yl)propyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine
4-[2-(piperidine-1-carbonyl)phenoxy]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
1-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(morpholin-4-yl)ethyl]acetamide
1-(4-benzylpiperidin-1-yl)-3-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]propan-1-one
1-(5-methyl-1,2-oxazole-4-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
2-[4-(7-methyl-1H-1,3-benzodiazol-2-yl)phenoxy]ethan-1-ol
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
(3R,4R)-4-cyclobutyl-3-methyl-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidin-4-ol
N-(diphenylmethyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
[(3R,4R)-1-(4-fluoro-2-methylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{[7-(adamantane-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
1-(carbamoylmethyl)-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
3-(3-fluorophenyl)-N-(2-hydroxyethyl)-N-(propan-2-yl)benzamide
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
1-(2-{[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}-4-methylpyrimidin-5-yl)ethan-1-one
1-[2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
5-{1-[3-(piperidin-1-yl)propanoyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-(adamantan-1-ylmethyl)-N-methylpropanamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}propanamide
N,N-dimethyl-3-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(piperidin-1-yl)piperidine
2-ethyl-5-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]pyrimidine
N-[(2R,3R)-1'-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
methyl 4-[2-(hydroxymethyl)pyridin-4-yl]benzoate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2,5-difluoro-N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
5-fluoro-8-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]quinoline
5-ethyl-N,2,3-trimethyl-N-[(2-methylpyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
4-[(diethylamino)methyl]-5-ethyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]furan-2-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 5-[(4-methoxy-4-methylpentan-2-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
4-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1λ6-thiane-1,1-dione
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methoxy-1H-indole-2-carboxamide
ethyl 1-[3-(1H-indol-3-yl)propanoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
4-[(6-chloropyridin-2-yl)methyl]-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-{[3-(methylsulfanyl)phenyl]methyl}propanamide
2,5-dimethyl-3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazine
1-[(2-fluorophenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-(2-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
[(2,3-dichlorophenyl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
(2E)-N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-fluorophenyl)prop-2-enamide
N-[2-(4-{[2-(3,5-difluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide