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4-[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]-3,3-dimethylpiperazin-2-one
(2E)-N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(4-fluorophenyl)prop-2-enamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(4-methylphenyl)methyl]amino}methyl)piperidin-2-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-1-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-cyclopropyl-N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3,5-dimethyl-4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-oxazole
9-(6-aminopyridine-3-carbonyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
4-(benzyloxy)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
(4aR,8aS)-6-(1-propylpiperidin-4-yl)-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2,3-difluoro-N-[2-(piperidin-1-yl)ethyl]benzamide
6-fluoro-4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-(1H-pyrazol-1-ylmethyl)piperidine-1-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(4-fluorophenyl)-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl]methylamine
9-(1,3-benzoxazol-2-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperidin-4-ol
methyl 6-[3-(2-chlorophenyl)pyrrolidin-1-yl]pyridine-3-carboxylate
2,5-dimethyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
4-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1-methyl-1,4,9-triazaspiro[5.5]undecane
2-{1-cyclohexyl-4-[(2,4,6-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
2-{4-[(2-methoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
(isoquinolin-5-ylmethyl)(methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
(4aS,8aR)-6-(2-ethyl-6-methylpyrimidin-4-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)acetamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
{[2-(furan-2-yl)phenyl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
1-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-3-(5-phenyl-1,3,4-thiadiazol-2-yl)urea
2-(2-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrrol-1-yl)pyridine
2-{4-[(3-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
1-{2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
1-[(2,3-difluorophenyl)methyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
3-(2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-cyclopropyl-6-(dimethylamino)-N-(1H-indol-5-ylmethyl)pyridine-3-carboxamide
6-(2-methoxyphenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(4-methoxyphenyl)methyl]-N,8-dimethyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(4aS,7aR)-1-(4-methoxybenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(morpholin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
1-{2-[2-(3-fluorophenyl)azepan-1-yl]-2-oxoethyl}pyrrolidin-2-one
1-(propan-2-yl)-5-(thiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
3-{1-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
4-{1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}thiomorpholine
2-{3-[(3-chlorophenyl)methyl]-5-[2-(1-methylpiperidin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-cyclopropyl-1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-4-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}pyridine
ethyl 1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)azepan-4-yl]piperidine-3-carboxylate
1-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(1H-indazol-1-yl)ethan-1-one