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methyl 2-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-yl)acetate
2-(2-aminoethyl)-N,N-bis(pyridin-3-ylmethyl)quinazolin-4-amine
N-methyl-5-{[methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amino]methyl}pyrimidin-2-amine
N4-methyl-N4-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]urea
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
1-(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-4H-1,2,4-triazole
3-methoxy-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydropyridin-2-one
3-[3-(4-fluorophenoxy)azetidine-1-carbonyl]piperidine-1-carboxamide
7-(2-ethoxypyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)benzamide
1'-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1,6-dimethyl-3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}methyl)-1H-1,3-benzodiazole
2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
2-(4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
3-chloro-4-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
3-{[butyl(methyl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
N-(2-methoxyethyl)-1-methyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-ethyl-4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(oxan-4-yl)-5-[5-(pyrrolidin-2-yl)thiophen-2-yl]-1H-1,2,4-triazole
2-[2-(3,4-dimethoxyphenyl)ethyl]-4-[4-(2-phenoxyacetyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-benzyl-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-(4-{2-[3-(morpholin-4-ylmethyl)phenoxy]ethyl}piperazin-1-yl)ethan-1-one
N,1-diethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
3-(3-methoxyphenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)propanamide
(4aS,8aR)-6-(1,3-benzothiazole-6-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
1-(4-fluorophenyl)-5-(methanesulfonylmethyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
3-({ethyl[(5-methylfuran-2-yl)methyl]amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methanesulfonyl-1,4-diazepane
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-methyl-1H-indole-4-carboxamide
{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
N3-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
3-methyl-7-[(3-phenoxyphenyl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
ethyl 3-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)piperidine-3-carboxylate
1-[3-(5-methylfuran-2-yl)butyl]-4-(pyridin-3-yl)piperidin-4-ol
4-{[4-(difluoromethoxy)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(hydroxymethyl)-1-[2-(2-methylphenyl)benzoyl]piperidin-3-ol
3-fluoro-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
3-(2-ethylphenoxy)-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]azetidine-1-carboxamide
2-{1-[ethyl(methyl)amino]propan-2-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-2-(2,2,2-trifluoro-1-phenylethoxy)ethan-1-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(6-methylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-6-(piperidin-4-yl)pyrimidin-4-amine