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1-[2-(1H-pyrazol-1-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(4-methoxyphenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]cyclopentane-1-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-1,2-dimethyl-1H-imidazole-4-sulfonamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]propanamide
5-(hydroxymethyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]furan-2-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(thiophen-2-yl)propan-1-one
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
1-[(3-methylpyridin-2-yl)methyl]-4-[3-(methylsulfanyl)propyl]piperazine
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-(4-hydroxy-2-methylphenyl)pyridine-3-carbonitrile
1-(5-methyl-1,2-oxazole-3-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
7-cyclohexyl-2-[5-(methoxymethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(1-{2-[(2,5-dimethylphenyl)carbamoyl]ethyl}-1H-imidazol-2-yl)benzoic acid
(1S,5R)-6-(1-phenyl-1H-pyrazole-4-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-1,3-diazinane-2,4-dione
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1,4-oxazepane
7-methyl-N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
4-{1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
(3R,4R)-3-cyclobutyl-4-methyl-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-3-ol
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-butyl-8-(2-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2,8-dimethyl-4-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]quinoline
6-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methyl-2,3-dihydropyridazin-3-one
3-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-1-(oxan-4-yl)urea
methyl (2S,4R)-1-methyl-4-[3-(1H-pyrazol-4-yl)benzamido]pyrrolidine-2-carboxylate
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(pyridin-2-yl)piperazine
4-(cyclopropylmethyl)-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-(3-acetyl-2-fluorophenyl)-2-[(furan-3-ylmethyl)(methyl)amino]acetic acid
2-[3-(pyridine-3-carbonyl)piperidin-1-yl]-4-(trifluoromethyl)pyrimidine
2-(1,3-benzoxazol-2-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
methyl (1R,3S,3aR,6aS)-1-butyl-5-ethyl-4,6-dioxo-3-(1,3-thiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-amino-8-(2-hydroxy-7-methylquinolin-3-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[(4-chlorophenyl)methyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-4-(thian-4-yl)piperazine
1-[(6-chloropyridin-2-yl)methyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-(3-phenoxypropyl)-1,3λ6,4-oxathiazinane-3,3-dione
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-6-yl]oxy}acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}propanamide
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
[(5-methoxy-1,3-benzoxazol-2-yl)methyl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
methyl({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(3-propylpyrrolidine-1-carbonyl)quinoline
3-(4-tert-butylbenzoyl)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[3-(pyridin-3-yl)propyl]butanamide
[7-(5-chloropyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(thiophen-2-yl)butanamide
3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-N-(4-methoxyphenyl)-3-oxopropanamide
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl][(1-methyl-1H-imidazol-5-yl)methyl]amine