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N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-methyl-4-{methyl[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-hydroxyethyl)-3-(piperidin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
1-(2-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)cyclopentan-1-ol
N-(3-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-3-methyl-1,2-oxazole-5-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(6-methyl-2-propylpyrimidin-4-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
1-ethyl-4-(2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-2,3-dihydro-1H-inden-2-yl)piperazine
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
1-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-(2-methanesulfonamidoethyl)urea
2-(1H-1,3-benzodiazol-1-yl)-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N2-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}pyrimidine-2,4-diamine
4-(2,3-dimethoxyphenyl)-2-methylquinazoline
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
5-{[4-(dimethylamino)azepan-1-yl]methyl}-2-hydroxybenzoic acid
1-[(4-fluorophenyl)methyl]-N-[3-(3-hydroxypiperidin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-chloro-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
2-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}benzonitrile
N-methyl-2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)pentanamide
2-({[(1-ethylpyrrolidin-2-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
1-(thiophen-2-yl)-2-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}amino)ethan-1-ol
ethyl 1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
5-{[4-(5-ethylfuran-2-yl)-1H-1,2,3-triazol-1-yl](phenyl)methyl}-1,3,4-thiadiazol-2-amine
6-ethyl-3-[1-(1H-imidazol-1-yl)butan-2-yl]-3,4-dihydroquinazolin-4-one
2-{1-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(furan-3-ylmethyl)-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-5-methoxy-4H-pyran-4-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3,5-dimethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-methyl-1-[2-(oxolan-2-ylmethoxy)phenyl]-3-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]urea
(3aR,6aS)-1-oxo-5-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(4-chloro-2-hydroxybenzoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
N-(cyclohexylmethyl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,4S)-1-[3-cyano-6-(propan-2-yl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-hydroxypropanamide
1-cyclopentyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
3-chloro-N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-1,2-oxazole-5-carboxamide
5-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]pyrazin-2-ol
dimethyl({3-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl})amine
5-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-N-(thiophen-3-ylmethyl)-1,3-thiazol-2-amine
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(3-fluoro-4-methoxyphenyl)methyl]-3-methoxy-2,2-dimethylpropanamide
9-[2-(2,5-dimethylphenyl)acetyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-phenyl-5-(thiophene-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(diethylamino)-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-[3-(4-tert-butylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(furan-2-yl)ethane-1,2-dione
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(oxane-4-carbonyl)piperazin-2-yl}ethan-1-ol
methyl (2S)-2-[(3-cyclopentaneamidophenyl)formamido]-2-cyclopropylacetate
5-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-tert-butyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-[(2-methylbutyl)amino]benzene-1-sulfonamide
6-fluoro-2-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline