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5-acetyl-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-hydroxy-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
5-methyl-3-[(2R)-pyrrolidin-2-ylmethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-[(2-fluorophenyl)methyl]piperidine
5-{2-[4-(5-ethylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
2-[1-cyclopentyl-4-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
1-(2-methoxyethyl)-6-oxo-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]piperidine-3-carboxamide
3-{1-[(3,5-difluorophenyl)methyl]piperidin-3-yl}-N-(3,5-dimethoxyphenyl)propanamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-[(4-methyl-1H-imidazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
3-methyl-8-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-2-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)-1H-indole
N,N-dimethyl-6-(3-phenoxypropyl)pyrimidin-4-amine
2-{[5-({[2-(3,5-dimethylphenoxy)ethyl](methyl)amino}methyl)pyrimidin-2-yl]amino}acetic acid
1-(2-{[1-(morpholin-4-yl)propan-2-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
3-{1-[(3-methoxyphenyl)methyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
5-ethyl-N4-methyl-N4-[(2-methylpyridin-4-yl)methyl]pyrimidine-2,4-diamine
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-fluoropyridine
3-ethyl-1-[2-fluoro-6-(trifluoromethyl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
(4aS,7aR)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)ethyl]piperidine-3-carboxamide
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(2-aminopyrimidin-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(diethylamino)ethyl]-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(pyridin-3-yl)propan-1-one
2-methoxy-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-{5-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-cyclopropylpropanamide
4-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
N-[4-(2-fluorophenoxy)phenyl]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-2-carboxamide
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinazolin-4-amine
2-[6-(2,6-dimethoxyphenyl)pyridin-3-yl]acetic acid
1-(3-methoxybenzoyl)-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
2-{[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]methyl}benzoic acid
methyl (2S)-2-{[2-(4-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-3-methylbutanoate
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-(methylsulfanyl)ethan-1-one
methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})(pyridin-3-ylmethyl)amine
N-[(4-hydroxyazepan-4-yl)methyl]-4-phenoxybenzene-1-sulfonamide
3-{1-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]piperidin-3-yl}-N,N-dimethylpropanamide
2-chloro-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}pyridine-4-carboxamide
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(quinolin-4-ylmethyl)amine
4-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
1-{2-methoxy-4-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
(2S)-2-(methoxymethyl)-1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidine
1-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
(3R,4R)-4-amino-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-ol
9-[(3,5-difluorophenyl)methyl]-6-oxa-9-azaspiro[4.5]decane
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3-acetamidopropanamide
N-[3-(2-methoxyphenoxy)propyl]-N-methylspiro[2.2]pentane-1-carboxamide