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N-methyl-4-{[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-1,3-thiazol-2-amine
2-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1,3-benzothiazole
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}oxane-4-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(1-phenylpiperidin-4-yl)acetamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
8-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R)-2-amino-4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pentanamide
6-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)pyridine-2-carboxylic acid
2-[3-(1-benzothiophen-3-yl)-4-methoxyphenyl]ethan-1-amine
N-butyl-N-(4-hydroxybutyl)-2-[N-(4-methylphenyl)methanesulfonamido]acetamide
4-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-phenyl-1H-pyrazole
(4aR,7aS)-1-acetyl-4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1H-imidazol-2-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]benzamide
3-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(2R)-2-hydroxy-3-methylbutanoyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl[3-(methylsulfanyl)butyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
(4aS,7aR)-1-[2-(5-fluoro-2-methylphenyl)acetyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(furan-2-yl)-3-phenyl-1-[3-(1H-pyrazol-1-yl)azetidin-1-yl]propan-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
N-ethyl-N-methyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetamide
3-methyl-1-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
2-(3-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}phenoxy)acetamide
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indazole-3-carboxamide
2-[3-benzyl-1-(4-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
1-cyclopentyl-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
8-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-[2-methoxy-5-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
3-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N,N-dimethylpropanamide
4-(1H-1,3-benzodiazol-1-yl)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
3-({[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}carbamoyl)benzoic acid
methyl (2S,4S)-4-(2-methoxybenzamido)-1-[(2-methylphenyl)methyl]pyrrolidine-2-carboxylate
4-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
2-(dimethylamino)-2-(3-methylphenyl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]acetamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)benzenesulfonamide
2-{3-cyclopentyl-5-[1-(propan-2-yloxy)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
9-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
{2-[(4-methoxypyrimidin-2-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
N-(2-tert-butylphenyl)-4-oxo-4-(1,2,3,6-tetrahydropyridin-1-yl)butanamide
(2R)-2-(methoxymethyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine
N-cyclopropyl-7-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyrimidin-2-amine
7-methyl-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,2-dihydroquinolin-2-one
{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazole
2-chloro-4-(1H-pyrazol-3-yl)benzoic acid
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyrimidin-2-ylmethyl)amine
N-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide