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N-ethyl-N-[(2-fluorophenyl)methyl]-1-methyl-1H-indazole-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)propanamide
1-cyclohexyl-N3,N5-dimethyl-4-oxo-N3-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-fluoro-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-sulfamoylbenzamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-{[5-(methoxymethyl)furan-2-yl]methyl}-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,5-dimethoxybenzamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-cyclopropyl-4-methylpyrimidine-5-carboxamide
4-(6-aminopyridine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
5-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(1-methylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylacetamide
1-[(5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}thiophen-2-yl)methyl]pyrrolidine
4-hydroxy-2-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-(3-fluorophenoxymethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-(2-aminopyrimidin-5-yl)-7-methoxy-N,N-dimethylquinoline-4-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
7-(pyridin-3-yl)-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-N,N-diethylaniline
2-(dimethylamino)-N-[3-({[(4-fluoro-3-methylphenyl)methyl]carbamoyl}amino)-2-methylphenyl]acetamide
1-{[4-(4-ethenylphenoxy)-3-methoxyphenyl]methyl}pyrrolidine
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
2-{1-cyclopentyl-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3R)-3-methyl-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazine
4-[(furan-3-ylmethyl)sulfamoyl]-N-(3-hydroxyphenyl)benzamide
7-(5-chloropyridin-2-yl)-4-(5-methyl-1,3-oxazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
4-(5,6-dimethylpyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[2-(dimethylamino)ethyl]amino}-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(1R,5R)-N,N-dimethyl-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-fluoro-2-[5-(oxolane-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
6-fluoro-2-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-cyclobutanecarbonyl-4-[4-(piperidin-3-yl)benzoyl]-1,4-diazepane
1-methyl-9-(prop-2-en-1-yl)-4-{thieno[2,3-d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-2-yl}pyridine
5,6-dimethyl-3-(thiomorpholine-4-carbonyl)-1,2-dihydropyridin-2-one
8-(2-methylpropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 7-oxo-3-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
(2S,4R)-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(3aR,5R,6S,7aS)-2-[2-methoxy-5-(propan-2-yl)benzenesulfonyl]-octahydro-1H-isoindole-5,6-diol
4-(1-benzyl-1H-imidazol-2-yl)-1-(5-methylthiophene-2-carbonyl)piperidine
N-tert-butyl-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]butanamide
(4aS,8aR)-6-(5-methyl-1,3-benzoxazol-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopentyl-4-[5-(morpholine-4-carbonyl)-1H-pyrrol-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(4-sulfamoylphenyl)ethyl]propanamide
6-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea