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7-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-amino-6-methylpyrimidin-4-yl)-4-[(2,6-dimethylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-2-[4-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1H-pyrazol-1-yl]acetamide
3-(2-methoxyethyl)-1-(2-methylpyridin-4-yl)piperidine-3-carboxylic acid
5-(4-fluorophenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-5-methyl-1H-pyrazol-1-yl]pyridine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-ethyl-5-methylpyrimidin-2-amine
N-[(3R,4R)-3-hydroxy-1-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
2-[1'-(2-methylbenzoyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
2-(4-chlorophenyl)-1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}ethan-1-one
2-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-methylpyrimidin-2-yl}phenol
(5R)-5-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
1-phenyl-3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
2-(furan-2-yl)-5-{1-[(4-methoxyphenyl)methyl]-1H-imidazol-2-yl}pyrimidine
N-(1-methyl-1H-1,3-benzodiazol-5-yl)-2-(pyrrolidin-3-yl)benzamide
1-acetyl-N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-1,2,3,4-tetrahydroquinoline-6-sulfonamide
3-[2-(aminomethyl)piperidine-1-carbonyl]-N-(1H-imidazol-2-ylmethyl)benzene-1-sulfonamide
1-(cyclohexylmethyl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-6-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
[1-(2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperidin-2-yl]methanol
N,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(1-methylpiperidin-4-yl)quinoline-4-carboxamide
4-(2-benzylmorpholine-4-carbonyl)pyridin-2-amine
1-[2-(pyrrolidin-3-yl)benzoyl]piperidine-4-carboxamide
3-[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]-2,2-dimethylpropan-1-ol
6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
2-(pyrimidin-2-ylsulfanyl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
N-[3-(2-methylpyrimidin-4-yl)phenyl]thiomorpholine-4-carboxamide
3-{[1-(4-methoxyphenyl)-5-phenyl-1H-pyrazol-3-yl]formamido}propanamide
8-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(pyrrolidin-1-yl)benzamide
methyl (1R,3S,3aR,6aS)-3-(1-benzofuran-2-yl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
1-(diethylamino)-3-[2-methoxy-5-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(methylsulfanyl)acetamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-(trifluoromethyl)benzamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-4,6-dimethylpyridine-3-carbonitrile
N-(1-hydroxypropan-2-yl)-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
N-{[(2S,4S)-1-(5-chlorothiophene-2-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}butane-1-sulfonamide
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(4-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
11-[(3-ethoxypropyl)amino]-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}azepane
N-butyl-N-methyl-3-{[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
methyl 2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]piperidine-1-carboxylate
2-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-5-methoxy-4H-pyran-4-one
ethyl 2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
3-{5-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
4-methyl-14-[3-(1H-pyrazol-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one