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N-cycloheptyl-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propanamide
N-[1-(4-chlorophenyl)ethyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
2-{1-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-ethyl-5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
3-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}imidazolidine-2,4-dione
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-azaspiro[5.5]undecan-9-amine
1-(2-ethoxyethyl)-N-[(3-hydroxyphenyl)methyl]-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-[2-(propan-2-yloxy)phenyl]pyridine-3-carboxamide
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-(dimethyl-1,3-thiazol-5-yl)acetamide
2-methoxy-N-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
2-{[4-phenyl-5-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-{2-oxo-2-[4-(pyridin-3-yl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
N3-(3-phenylprop-2-yn-1-yl)-N3-propylpiperidine-1,3-dicarboxamide
4-(4-methoxybutyl)-N-[1-(1-phenylethyl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(pyridin-3-yl)propanoyl]pyrrolidine-2-carboxamide
7-chloro-3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
3-[(3R,4S)-1-(2,6-diaminopyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2R,3R,6R)-5-(2-ethylpyrimidine-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{3-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}acetamide
2-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1,7-dimethyl-1H-indole
N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-(5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
9-[4-(1H-imidazol-1-yl)butanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(diethylamino)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-phenylpyrrolidin-2-one
4-({3-[1-(pyridin-4-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)morpholine
3-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
4-(5-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
1-{5-[(cyclopropylamino)methyl]-2-methoxyphenoxy}-3-(piperidin-1-yl)propan-2-ol
(2S,4S)-4-amino-1-(7-chloro-1-methyl-1H-indole-2-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-(2-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-5-yl)acetamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]morpholine-2-carboxamide
4-(4-ethyl-5-methylthiophene-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
3-methyl-N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]but-2-enamide
1-(1,2-oxazole-3-carbonyl)-3-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N,1,3-trimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
4-{4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine-1-carbonyl}morpholine
6-(2,5-dimethylfuran-3-yl)-N-(1-methoxybutan-2-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-yl)ethan-1-ol
1-[(2S,4R)-1-[(4-phenylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
5-({[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(8-methoxyquinolin-5-yl)methyl]methylamine
5-(azocane-1-carbonyl)-N-butyl-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide