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methyl 3-[(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]propanoate
2-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol
5-[4-phenyl-5-(2,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]pentan-1-amine
5-[5-(2-methylpropyl)-1,2-oxazol-3-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2-{2-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}propan-1-one
1-methyl-4-({5-[5-(4-methylphenyl)-1H-pyrazol-3-yl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
3-hydroxy-N-[2-(2-methylpropoxy)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
N-cyclopropyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(1S,5S)-3-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(2R,3R)-3-amino-1'-[(3-hydroxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[(2-hydroxyethyl)(1,3-thiazol-2-ylmethyl)amino]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
4-(2,3-dichlorophenyl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-1,2,3-triazole
6-(2-aminoethyl)-N-cyclopropyl-N-(thiophen-3-ylmethyl)pyrimidin-4-amine
4-({[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
3-(1-cyclopropanecarbonylpiperidin-3-yl)-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
2-(4-methylpyridine-3-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2S)-1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-methyl-2-phenylpiperazine
(2S,4S)-4-amino-1-(isoquinoline-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
3-(3-fluorophenyl)-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-pyrazole-4-carboxamide
methyl 1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine-2-carboxylate
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(pyridine-4-carbonyl)piperidine-4-carboxylic acid
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-tert-butyl-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
1-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-3-ol
1-(carbamoylmethyl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}piperidine-3-carboxamide
4-(1H-indol-3-yl)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
4-(5-fluoro-2-methylphenyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methanesulfonyl-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
4-(4-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-ethyl-4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amine
5-(4-methylphenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-3-carboxamide
2-[2-(dimethylamino)ethyl]-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-1-(propan-2-yl)-4-[2-(pyrrolidin-1-yl)benzoyl]piperazine
1-(2-methoxyethyl)-4-{[4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}piperidine
2-methyl-6-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
7-(cyclopropylmethyl)-2-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(4,4-difluoropiperidin-1-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
3-{5-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[2-(2-methanesulfonamidopropanamido)-4-methylphenyl]pentanamide
N-(cyclopropylmethyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
2-chloro-6-methoxy-4-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}phenol
methyl 2-[({3-[(2,3-difluorophenyl)carbamoyl]phenyl}methyl)(methyl)amino]acetate
(4R)-1-{3-[(2-chloro-6-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-4,7,7-trimethyl-2-oxabicyclo[2.2.1]heptan-3-one