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(2S,4R)-4-amino-1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-2,4-dimethylpyrimidine-5-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
2-(4-{[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-1-yl)pyrimidine
1-ethyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
N-{2-[(1R,7S)-6-(azocane-1-carbonyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]ethyl}acetamide
2-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}morpholin-2-yl)ethan-1-amine
(2R,3R)-3-amino-1'-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aS,8aR)-1-(2-aminoethyl)-6-(1-methylcyclohexanecarbonyl)-decahydro-1,6-naphthyridin-2-one
N-ethyl-1-[2-(3-fluorophenyl)ethyl]-N-(2-hydroxyethyl)-6-oxopiperidine-3-carboxamide
4-(3-ethyl-1H-pyrazole-4-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
2-[3-(dimethylamino)propyl]-9-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-2-[(4-methylphenyl)amino]-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
N-ethyl-N-[(4-fluorophenyl)methyl]-3-(4-hydroxyphenyl)propanamide
3-(2-{2-[1-(propan-2-yl)-2,3-dihydro-1H-indol-5-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazolidin-2-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N,2-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
7-methoxy-N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-[2-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)-4-(thiophen-3-yl)phenoxy]acetic acid
5-(4-tert-butylbenzoyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3-fluorophenyl)-3-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(ethoxymethyl)-1-methyl-5-(5-methylthiophen-2-yl)-1H-1,2,4-triazole
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-[2-(dimethylamino)ethyl]-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
1-methyl-2-{1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazol-2-yl}-1H-imidazole
(1R,5S)-8-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3,8-diazabicyclo[3.2.1]octane
1,4,6-trimethyl-3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
1-(3-hydroxypropyl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
4-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N,N-dimethyl-4-[2-(phenylamino)pyrimidine-5-carbonyl]piperazine-1-carboxamide
2-(2,5-dimethylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
2-(4-butyl-2,3-dioxopiperazin-1-yl)-2-phenyl-N-(1,3-thiazol-2-ylmethyl)acetamide
N-(2-hydroxyethyl)-5-[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
[(3S,7S)-5-[4-(trifluoromethyl)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
(1S,3R)-3-amino-N-[(2-methoxyphenyl)methyl]-N-(3-methoxypropyl)cyclopentane-1-carboxamide
2,3,5,6-tetramethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}benzamide
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-indole
N-(3-ethylphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
(4aS,8aR)-6-(5-ethoxyfuran-2-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-ethyl-5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyrimidin-2-amine
3-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-2-(cyclopentylmethyl)-6-methyl-1-(pyridin-3-ylmethyl)-1,4-dihydropyridin-4-one
2-{2-[3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
3-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}benzonitrile
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(1H-pyrazole-4-carbonyl)piperazine
N-(2-hydroxypropyl)-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
5-chloro-3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one