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3-{1-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-4-yl}phenol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(2-methylphenyl)piperidine
3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]-N-(furan-2-ylmethyl)propanamide
3-[2-(dimethylamino)ethyl]-8-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-methylphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-5-(pyrimidin-5-yl)pyrimidin-2-amine
2-[4-(7-fluoroquinazolin-4-yl)piperazin-1-yl]-1-(morpholin-4-yl)ethan-1-one
8-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{[1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
(1S,5R)-3-[3-(1,3-benzothiazol-2-yl)propanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(2-ethylphenoxy)ethyl]-2-fluoro-6-hydroxy-N-methylbenzamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
3-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
7-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-2,4-dimethylquinoline
1-(1-benzylpiperidin-4-yl)-N-(oxan-4-yl)piperidine-3-carboxamide
(3R,4S)-4-[4-(furan-3-ylmethyl)-1,4-diazepan-1-yl]oxolan-3-ol
2-{[4-(3-methoxyphenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-acetyl-N-{2-[methyl(phenyl)amino]ethyl}piperidine-3-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,7S)-6-(4-methyl-3-oxopiperazine-1-carbonyl)-3-[(3-methylphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
ethyl 1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
1-(2-methoxyphenyl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-methyl-4-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,4-dihydroquinoline-3-carboxamide
2-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
3-{[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}azepan-2-one
6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-[(2R)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-(2-methanesulfonylethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-benzyl-2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-3-(3-hydroxy-3-methylbutyl)benzamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
(2S,4S)-4-(4-{2-[(5-fluoro-2-methylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
(2S,4S)-N-ethyl-4-(3-hydroxypropanamido)-1-[(1-methyl-1H-indol-6-yl)methyl]pyrrolidine-2-carboxamide
1-(3-{2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}phenyl)imidazolidin-2-one
2-[2-(dimethylamino)ethyl]-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
3-(2-hydroxyphenyl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-1H-pyrazole-5-carboxamide
methyl (1S,3S,3aR,6aS)-5-ethyl-3-(1-ethyl-1H-imidazol-5-yl)-1-(hydroxymethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2,6-dimethoxy-N-methylpyridine-3-carboxamide
N-[2-(3-chlorophenyl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-2,4-dioxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-(morpholin-4-ylmethyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
3-methyl-N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
1-[1-(2-hydroxyethyl)piperidine-4-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1H-indol-4-ylmethyl)-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-{3-cyclohexyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-imidazol-1-yl)-6-methylpyridine
1-(5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
3-{4-[4-methoxy-4-(prop-2-en-1-yl)piperidin-1-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
2-(azepan-1-yl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
1-{4-[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-{2-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide