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6-(piperazin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
ethyl[(4-methanesulfonylphenyl)methyl]{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(5-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-1-(thiomorpholin-4-yl)ethan-1-one
3-butyl-1-methyl-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperazin-2-one
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
(1S,2R)-N1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
4-methoxy-3-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}phenol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(dimethylamino)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]-2-(3-methylphenyl)acetamide
(5-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-1H-1,3-benzodiazol-2-yl)methanol
4-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-N-(5-methylpyridin-3-yl)benzamide
2-[3-({9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)phenoxy]acetamide
2-(2,3-dimethoxyphenyl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
2-(2,2-dimethylpropanamido)-N,5-dimethyl-N-(1H-pyrazol-5-ylmethyl)thiophene-3-carboxamide
N-(furan-2-ylmethyl)-4-(morpholin-4-yl)-N-(pyridin-2-ylmethyl)butanamide
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
methyl 1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-imidazole-4-carboxylate
4-{[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]methyl}-N-methylbenzamide
3-{2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]ethyl}-1,3-oxazinan-2-one
N-[(3S,4R)-1-(5-methyl-2-phenylfuran-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
2-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-2-[methyl(pyridin-3-ylmethyl)amino]acetic acid
7-chloro-4-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]quinoline
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-fluorophenyl)methyl]piperidine-3,5-dicarboxamide
1-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1H-pyrazole-5-carboxamide
3-{1-[1-(thiophene-3-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
(1S,5R)-N-(2-ethylphenyl)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-benzyl-4-(4-chloro-2-fluorobenzoyl)piperazin-2-one
5-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
methyl (1R,3S,3aR,6aS)-5-ethyl-3-(2-fluoro-3-methoxyphenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-cyclopropyl-6-oxo-N-[(1-phenylcyclohexyl)methyl]piperidine-3-carboxamide
4,4,4-trifluoro-1-(4-phenyl-1,4-diazepan-1-yl)butan-1-one
6-ethoxy-2-{1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}quinoline
1-(1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)pyrrolidin-2-one
(3aS,7aR)-2-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(2-phenylpropan-2-yl)amino]methyl}piperidin-2-one
2-(3-chloro-4-fluorophenyl)-2-[4-(pyridin-3-yloxy)piperidin-1-yl]acetic acid
4-[(2-chlorophenyl)methyl]-1-[2-(dimethylamino)benzoyl]-1,4-diazepan-5-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-cyclobutyl-2-[4-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)morpholin-3-yl]acetamide
5-[methyl(2-phenylethyl)amino]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
1-cyclohexyl-4-[1-(methylsulfanyl)propan-2-yl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide