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3-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-indole
3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]urea
[5-(1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-phenyl-1H-imidazol-5-yl)furan-2-yl]methanol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-ethyl-1,3-oxazole-4-carboxamide
1-[4-(cyclopropylmethyl)piperazin-1-yl]-3-(4-methoxyphenyl)-3-phenylpropan-1-one
2-(4-{[(2-chloro-4-fluorophenyl)carbamoyl]amino}piperidin-1-yl)-N-cyclopropylacetamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]ethan-1-ol
N-(isoquinolin-5-ylmethyl)-N,3-dimethylthiophene-2-carboxamide
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
methyl({2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})(3-phenylpropyl)amine
8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
[(3R,5R)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
propan-2-yl 4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-(2,3-dimethoxyphenyl)-2-methyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-[2-methoxy-4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)furan-2-carboxamide
1-[5-(4,4-difluoropiperidine-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
(3aS,7aR)-2-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-(dimethylamino)-2-(4-methylphenyl)-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethan-1-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}benzoic acid
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-phenylpiperidin-3-amine
N-(2-methoxy-5-phenylphenyl)-2-(methoxymethyl)piperidine-1-carboxamide
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
2-methyl-5-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidine-1-carbonyl)pyrazine
1-phenyl-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(8R,9aS)-8-hydroxy-2-(1H-indol-2-ylmethyl)-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
2-(3-methoxyphenyl)-5-(oxolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl 3-{[1-(cyclopropylmethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
3-[4-({methyl[(5-methylthiophen-2-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
1-benzyl-4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]pyrrolidin-2-one
1-(3-methylbutyl)-3-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-({7-[5-(methoxymethyl)furan-2-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-1-[1-(6-methylpyridin-3-yl)ethyl]urea
8-(1-acetylpiperidine-4-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(pyrazin-2-ylmethyl)pyridin-2-amine
3,3-dimethyl-1-[(3S,4R)-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-chromen-4-one
(2R,3R,6R)-3-phenyl-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-N,N-dimethylpyrrolidin-3-amine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
4-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-(3-methylphenoxy)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}azetidine
1-(diethylamino)-3-[5-({[(3,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one