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2-{5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
(2S,4S,5R)-2-ethyl-4-[ethyl(methyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
5-{[benzyl(methyl)amino]methyl}-N-ethyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
8-[(2-chloro-6-fluorophenyl)methyl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,2S)-2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}cyclopentan-1-ol
N-[3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}methoxy)phenyl]propanamide
(3S,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
2-(1-propylpiperidin-4-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-(3-hydroxypropyl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxamide
{4-[2-methyl-2-(morpholin-4-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
N-[1-(4-methanesulfonylphenyl)propyl]cyclopentanamine
2-cyclopentyl-1-[9-(morpholin-4-yl)-3-azaspiro[5.5]undecan-3-yl]ethan-1-one
methyl (2S)-2-{[4-(1H-pyrazol-5-yl)phenyl]formamido}propanoate
1-[3-oxo-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propyl]piperidin-2-one
1-methyl-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
3-[1-(5-ethoxyfuran-2-carbonyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}thiophene-2-carboxamide
2-[4-(4,6-dimethylquinolin-2-yl)piperazin-1-yl]-N-(propan-2-yl)acetamide
N-(1,3-dihydroxypropan-2-yl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
8-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-(4-fluorophenyl)-4-[1-(oxan-4-yl)piperidin-3-yl]piperazine
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methoxybenzene-1-sulfonamide
(1R,2S,9R)-11-[(1-phenyl-1H-pyrazol-5-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(dimethylamino)-4-methyl-N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]pyrimidine-5-carboxamide
5-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]-2-ethylpyrimidine
1-[(3,4-dimethylphenyl)methyl]-4-[2-(3-methoxyphenoxy)acetyl]piperazin-2-one
4-(1H-indazol-6-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
6-(2-chlorophenyl)-7-methyl-8-oxo-N-(pentan-3-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-amino-4-(4-hydroxy-3-methylphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
ethyl 2-chloro-5-({[(1S,2S)-2-hydroxycyclohexyl]carbamoyl}amino)benzoate
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-[2-(pyridin-4-yl)ethyl]benzamide
3-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
2-hydroxy-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(3-hydroxypropanoyl)pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
N-[2-(diethylamino)ethyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
(1R,5R)-6-(2,4-difluorobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(oxolan-3-yl)-5-[4-(pyrrolidin-1-yl)phenyl]-1,2,4-oxadiazole
4-hydroxy-N-methyl-N-[3-(2-methylphenoxy)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[2-(1,2-benzoxazol-3-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propyl)pyrrolidin-2-one
N-ethyl-5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-amine
(2S,4S)-N,N-diethyl-1-(naphthalen-1-ylmethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
(2R,4S)-1-(2H-1,3-benzodioxol-4-ylmethyl)-4-hydroxypiperidine-2-carboxylic acid
2-(but-3-enoyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide