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2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(dimethylamino)ethyl]acetamide
2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}pyridine-3-carboxylic acid
N-[(2-ethoxy-3-methoxyphenyl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
{[2-(cyclopentyloxy)phenyl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
3-(1,2-oxazinan-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
4-(azocan-1-yl)-N-(1-methoxypropan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-(5-chloro-2-methoxyphenyl)propanamide
5-{1-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1H-imidazol-2-yl}quinoline
3-methyl-8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-methoxyethan-1-one
9-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-6-oxo-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}piperidine-3-carboxamide
{4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]phenyl}methanol
1-ethyl-4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
3-(1,3-benzothiazol-2-yl)-1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}propan-1-one
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
4-(cyclopropylmethyl)-1-(2,3-dimethyl-1H-indole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-[1-(cyclohexylmethyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-{1-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}methanesulfonamide
2-(3-phenylpropyl)-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
methyl[(1-methyl-1H-imidazol-2-yl)methyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
(3S,4R)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-{[3-(dimethylamino)phenyl]methyl}-3-(2,5-dioxoimidazolidin-4-yl)propanamide
N-[(3R,4R)-3-hydroxy-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl]pyrazine-2-carboxamide
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
9-methoxy-7-(4-methoxyphenyl)-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(butan-2-yl)-2-ethyl-4-methyl-N-[(4-methylphenyl)methyl]-1,3-oxazole-5-carboxamide
4-({1-benzyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)morpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
6-butyl-2-(4-{[ethyl(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methylpyridin-2-amine
3-(4-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}phenyl)prop-2-yn-1-ol
(3R)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-ol
2-benzyl-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecane
4-(2-ethylpyrimidine-5-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-cyclopentyl-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-(3-methoxyphenyl)-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methyl-5-(trifluoromethyl)benzamide
6-(4-methoxyphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
2-(3-cyano-2-methyl-1H-indol-1-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}acetamide
5-[(benzyloxy)methyl]-3-cyclopropyl-1-(4-methanesulfonylphenyl)-1H-1,2,4-triazole