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1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(3,4-dimethyl-1H-pyrazol-5-yl)propan-1-one
5-(2-{4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
9-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
6-methyl-5-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methoxy-1-methyl-1H-indole
1-(4-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
4-(1H-imidazol-1-yl)-1-[(2E)-4-methylpent-2-en-1-yl]piperidine-4-carboxylic acid
1-cyclohexanecarbonyl-N,N-bis(prop-2-en-1-yl)pyrrolidine-2-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidin-3-ol
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-(2-methoxy-4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
1-methyl-1'-[3-(pyridin-3-yl)propyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[(1-ethylpiperidin-3-yl)methyl]-N-methylthian-4-amine
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(3R,4S)-4-(propan-2-yl)-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]acetamide
3-({1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
2-ethyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]cyclopentane-1,3-dicarboxamide
N-[2-(2-chlorophenoxy)ethyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
5-methyl-N-[3-(pyridin-3-yloxy)propyl]-1-benzofuran-2-carboxamide
4-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(cyclopentylmethyl)-6-methyl-3-(4-methylpiperazine-1-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-dihydropyridin-4-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(pyridin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-(4-methoxyphenyl)-1-phenyl-1H-pyrazole
1-[(3-methylpyridin-2-yl)methyl]-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazine
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-methyl-1-benzofuran-5-carboxamide
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methoxy-2-methylpropan-1-one
(1r,4r)-4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-amido)cyclohexane-1-carboxylic acid
2-[3-(3-fluorophenyl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-ethyl-3-{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3aS,6aS)-5-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-octahydropyrrolo[3,4-b]pyrrol-1-yl]-2-methoxyethan-1-one
1-{1-ethyl-5-[(4-methoxy-2,5-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-(1,2-benzoxazol-3-yl)-N-[(5-oxo-1-phenylpyrrolidin-3-yl)methyl]acetamide
N-{2-[5-(2,1,3-benzoxadiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}propanamide
6-(4-chlorophenyl)-N-(2-methoxy-2-methylpropyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2R)-2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-2-phenylethan-1-ol
6-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
1-(3,3-diphenylpiperidin-1-yl)-2-(pyridin-3-yl)ethan-1-one
3-{[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,2,3-trimethylbut-3-en-1-one
1-(1-{1-[(2E,4E)-5-(4-fluorophenyl)penta-2,4-dien-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-chloro-N-(2-methoxyethyl)-4-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperidin-2-yl)ethan-1-ol
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl){[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine