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(1S,5R)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-cyclopropyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]pyrimidine-5-carboxamide
4-(3-{[(dimethyl-1,2-oxazol-4-yl)methyl]amino}butyl)-2-methoxyphenol
N-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
(3R,4S)-4-cyclopropyl-1-{3-[4-(2-methylpropoxy)phenyl]-1H-pyrazole-5-carbonyl}pyrrolidin-3-amine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
1-{1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}azepan-4-ol
N-ethyl-2-(3-methanesulfonamidopropanamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
4-acetyl-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}piperazine-1-carboxamide
2-(adamantan-1-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
7-(6-chloro-8-methylquinolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
N-butyl-N-(furan-2-ylmethyl)-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(1S,5R)-6-benzyl-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-4-carbonitrile
N-cycloheptyl-4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carboxamide
6-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
3-methyl-2-{5-[3-(1H-pyrazol-4-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridine
9-(cyclopropylmethyl)-1-methyl-4-(2-methylbenzoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(morpholin-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylbenzamide
7-{4-[1-(dimethylamino)ethyl]phenyl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
1-[ethyl(methyl)sulfamoyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl]propanoic acid
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
3-ethyl-1-(5-methyl-4-phenylthiophene-3-carbonyl)piperidine-3-carboxylic acid
(2S)-2-amino-3-cyclohexyl-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
N-cyclopentyl-3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(morpholine-2-carbonyl)-8-azabicyclo[3.2.1]octane
2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1,3-thiazole-4-carboxamide
6-{3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
methyl 4-(4-{[2-(2-acetamidoethyl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
3-(3-methoxyphenoxy)-1-(2-methylfuran-3-carbonyl)azetidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)propan-1-one
N-[4-(piperidine-1-carbonyl)phenyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-[(3R)-1-benzylpyrrolidin-3-yl]-3-methyl-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
3-(2-fluorophenyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazole
methyl 5-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-chloro-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1R,6S)-3-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
3-methyl-1-[1-(6-{[2-(pyridin-3-yl)ethyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
5-(azepane-1-carbonyl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxy-6-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(diethylamino)-3-{2-methoxy-4-[({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)methyl]phenoxy}propan-2-ol
1-{[5-(4-fluorophenyl)furan-2-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
2-(4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}phenyl)ethan-1-amine
4-oxo-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,4-dihydroquinoline-2-carboxamide
3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile