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N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
8-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-methoxy-1-{4-[4-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
N-(2,4-dimethoxyphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]benzonitrile
1,3-dimethyl-N-(4-phenylbutyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
[(4S)-4-amino-5-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-5-oxopentyl]urea
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-4-(hydroxymethyl)benzamide
(2S)-3-(4-hydroxyphenyl)-2-{[3-(4-methylphenyl)-1H-pyrazol-5-yl]formamido}propanamide
1-methyl-2-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-imidazol-2-yl)-1H-imidazole
5-acetyl-N-(2-methoxyethyl)-2,4-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrrole-3-carboxamide
4-(benzyloxy)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
6-ethyl-2-methyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]quinoline-4-carboxamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
4-(4-chlorophenyl)-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
1-[3-(4-propylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
(1S,9R)-11-[6-(piperidin-4-yl)pyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-[(4-chlorophenyl)methyl]-8-{[(2R)-1-methylpyrrolidin-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]-3,9-diazaspiro[5.6]dodecan-10-one
9-(6-cyclopropylpyrimidin-4-yl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
N-cyclobutyl-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-methoxyphenyl)-3-methyl-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperazin-2-one
N-butyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-ethyl-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidine-3-carboxylic acid
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)[2-(4H-1,2,4-triazol-4-yl)ethyl]amine
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
1-ethyl-3,5-dimethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-pyrazole-4-carboxamide
1-[2-(4-tert-butylphenoxymethyl)-4-hydroxypyrimidine-5-carbonyl]-2-methyl-1,4-diazepan-5-one
3-(4-chlorophenyl)-2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-[2-(piperidin-1-yl)ethyl]propanamide
1-methyl-6-(propan-2-yl)-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-methyl-6-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyridazine
4-[4-(diphenylmethyl)piperazine-1-carbonyl]imidazolidin-2-one
1-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
9-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-indole-6-carboxamide
2-benzyl-N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-3-oxopiperazine-1-carboxamide
3-(4-methyl-1H-pyrazol-1-yl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]thiophene-2-carboxylic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
propyl (4aR,7aS)-4-(1-methyl-1H-pyrazole-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-{[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-(2-methyloxane-2-carbonyl)-4-(2-phenoxyethyl)piperazine
1-(1-{6-[4-(hydroxymethyl)piperidin-1-yl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one