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(3aR,7aS)-2-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-ethyl-N-[1-(4-methylphenyl)cyclopropyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-butyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
(3S,4R)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N2-benzyl-6-(thiophen-3-yl)-1,3,5-triazine-2,4-diamine
N-methyl-N-(2-methylprop-2-en-1-yl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
4-(3-hydroxy-3-methylbutyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide
N-[2-(benzylsulfanyl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-cyclopropyl-1-phenyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
N-(3-chloro-4-methoxyphenyl)-6-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
N-ethyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4-methylpentan-2-yl)({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methylquinolin-4-yl)pyrrolidin-3-yl]methanol
(2S,4S)-4-amino-1-(2-aminopyridine-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
(3S,4S)-N-(2-benzylphenyl)-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
5-ethyl-N4-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]pyrimidine-2,4-diamine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(1R,5R)-N,N-dimethyl-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]azocane
1-{2-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3-benzotriazole
3-[4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-benzyl-N-methylpropanamide
7-[(2-fluorophenyl)methyl]-2-[3-(1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,4-dimethylpyrimidin-2-amine
1-(4-methoxyphenyl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazin-2-one
1-methyl-N-{2-[methyl(phenyl)amino]ethyl}-1H-1,3-benzodiazole-5-carboxamide
1-{5-[(3,5-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
(4aR,7aS)-1-(pyrimidin-2-yl)-4-[2-(pyrrolidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-[ethyl(methyl)amino]ethan-1-one
8-fluoro-2-({[4-(oxolan-2-yl)butyl]amino}methyl)quinolin-4-ol
methyl 3-(2-methyl-1,3-thiazole-4-carbonyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{[1-(2-hydroxybutyl)-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
N-{2-[1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-4-yl]ethyl}acetamide
4-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane
(1S,5R)-6-(cyclobutylmethyl)-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-5-phenoxyfuran-2-carboxamide
2-oxo-8-[(thiophen-2-ylmethyl)carbamoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(1S,5R)-3-{[4-(methylsulfanyl)phenyl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-ethyl-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[4-hydroxy-1-(thiophen-3-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
1-cyclobutyl-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-3-ol
N-{1-[2-(dimethylamino)ethyl]piperidin-4-yl}-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole