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7-methyl-2-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
2-[3-(2-methylphenoxy)azetidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
7-[2-(1H-indol-3-yl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(1,3-dihydro-2-benzofuran-5-yl)-2-(3-fluorophenyl)azepane-1-carboxamide
2-{1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-2-yl}pyridine
3-(2,3-dihydro-1H-inden-5-yl)-1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methylurea
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
6-[(3S,4R)-3-cyclopropyl-4-(oxane-4-amido)pyrrolidin-1-yl]pyrazine-2-carboxamide
5-ethyl-2-methyl-4-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
1-[1'-(2-ethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-methyl-7-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(prop-2-en-1-yl)benzamide
1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carboxamide
(2R,3S,6R)-5-(6-methylpyridazin-3-yl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(benzyloxy)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-{2-[7-(3-chlorothiophene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
1-cyclohexyl-N-[(3,4-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-3-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}propanamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
(3E)-1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)hex-3-en-1-one
1-methyl-N-[(4-phenyloxan-4-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methoxyphenol
(1S,5R)-6-(5-methoxyfuran-2-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-methyl-9-(thiophene-2-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
1-ethyl-8-(1-hydroxypropan-2-yl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-(cyclopropylmethyl)-1-(oxane-4-carbonyl)piperidine-3-carboxylic acid
3-{1-oxaspiro[4.4]nonan-3-yl}-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
1-(4-fluorophenyl)-4-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]butane-1,4-dione
ethyl 1-(1H-imidazol-2-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(2S)-2-amino-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methyl-3-phenylpropan-1-one
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-phenylpiperazine
4-[2-(1-phenylethyl)-1H-imidazol-1-yl]benzamide
2-(2-hydroxyethyl)-6-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
methyl 2-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]benzoate
4-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-1-(3-methoxyphenyl)pyrrolidin-2-one
6-(2,5-dimethylfuran-3-yl)-2-{4-[(3-methoxypiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
N-(2-hydroxy-2-phenylethyl)-4-(propylsulfamoyl)benzamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[2-methyl-2-(piperidin-1-yl)propyl]pyrrolidin-3-ol
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)pyrrolidine-2,5-dione
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
1-ethyl-3-(pyrrolidine-1-carbonyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,5R)-N-(3-chloro-4-fluorophenyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide