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{[(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(2S,4R)-4-[4-({[(3-chloro-2-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-hydroxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-{[1-(3-chloro-4-fluorobenzenesulfonyl)piperidin-3-yl]methyl}pyridine-3-carboxamide
2-chloro-5-{5-[(2,5-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
1-[(2,4-dimethoxyphenyl)methyl]-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
1-{5H,6H-imidazo[2,1-b][1,3]thiazole-3-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-(4-hexylphenyl)-4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carboxamide
(2S)-1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
5-{3-carboxy-5-[(propan-2-yl)sulfamoyl]phenyl}thiophene-2-carboxylic acid
ethyl 2-{2-[(7-chloro-3,5-dimethyl-1-benzofuran-2-yl)formamido]ethyl}-1,3-thiazole-4-carboxylate
(4aR,7aS)-1-[2-({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-methylphenyl)propan-2-yl]-3-(methylsulfanyl)propanamide
N-[2-methyl-5-({methyl[3-(oxolan-2-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
3-phenyl-1-[1-(piperidin-4-yl)piperidin-3-yl]propan-1-one
7-(3-chlorophenyl)-4-(dimethyl-1,3-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
1-[2-methyl-5-oxo-4-(3-phenylphenyl)piperazine-1-carbonyl]cyclopropane-1-carboxamide
N-cyclopropyl-4-(3,5-difluoro-2-methoxyphenyl)benzamide
N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-(piperidin-4-yl)pyrimidin-4-amine
N-cyclooctyl-1-(2-methoxyethyl)-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-methyl-8-(1,3-thiazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(pyridin-4-yl)propan-1-one
4-[(6-ethoxypyridin-3-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
methyl 4-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}benzoate
N-(2-methoxyethyl)-1-{1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
1-(oxolane-2-carbonyl)-4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepane
3-(1-ethyl-1H-imidazol-2-yl)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidine
N-[2-(2-oxopiperidin-1-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S,5R)-4-{[2-(dimethylamino)ethyl]carbamoyl}-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
2-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)-1,2-oxazinane
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
(3-{2-[1-(4-chloro-3-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-ethyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-2-methoxypyridine
2-methoxy-1-(1'-{spiro[2.3]hexane-1-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(3aS,6aS)-2-methanesulfonyl-5-(propane-2-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-chloro-5-(methylcarbamoyl)phenyl]-4-(2-methoxyethyl)piperazine-1-carboxamide
2-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}-N-[(2-fluorophenyl)methyl]acetamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}cyclopropanamine
{[4-cyclopropyl-5-(1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
ethyl 4-{4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}piperidine-1-carboxylate