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6-amino-N-({1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
3-[5-(5-chlorothiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-methyl-1'-(pyrazine-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-{1-[(1-ethyl-1H-indol-6-yl)methyl]piperidin-4-yl}-N-methylacetamide
2-(1H-1,3-benzodiazol-1-yl)-N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]acetamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-methoxy-3-(2,4,6-trimethylphenyl)pyrazine
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-1,2,5-thiadiazole-3-carboxamide
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
5-methyl-3-phenyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-4-carboxamide
1-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)-3-methylimidazolidin-2-one
1-[(2-chlorophenyl)methyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
{3-benzyl-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-3-yl}methanol
N-(3-methoxypropyl)-6-methyl-2-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)quinazolin-4-amine
[(3,5-dimethoxyphenyl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
5-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-chloro-N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-methyl-4-({5-[(E)-2-phenylethenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-{[3-(trifluoromethyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
2-methoxy-3-(3,4,5-trimethoxyphenyl)pyrazine
(2R,6R)-11-methoxy-4-(3,3,3-trifluoropropyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-fluoro-2-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
(3S)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
3-[(4aR,7aS)-4-{[3-(methylsulfanyl)phenyl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-hydroxy-3-({[(2-methylpyridin-4-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
(1S,5R)-6-benzyl-3-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[4-(piperidine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}piperidin-4-ol
(2S,4S,5R)-4-[ethyl(pyridin-4-ylmethyl)carbamoyl]-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
1-[2-(furan-2-yl)azepan-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
[7-(3-fluoro-4-methoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzene-1-sulfonamide
5-{[benzyl(methyl)amino]methyl}-N-(2-hydroxypropyl)-1,2-oxazole-3-carboxamide
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]butan-1-one
1-cyclopentyl-4-{[methyl({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})amino]methyl}pyrrolidin-2-one
1-(2-fluoro-4-methoxyphenyl)-3-methyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]urea
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
6-methoxy-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-(5-methylfuran-2-yl)benzoyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
1-[(4aR,8aR)-4a-hydroxy-7-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[2-(1H-indol-4-yl)pyridin-3-yl]-2-methylpropanamide
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
1-[(3,5-dichloro-4-methylphenyl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-(2-methoxy-4-{[methyl(2-methylpropyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
2-(4-fluoro-2-methoxyphenyl)-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]acetic acid
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-[(2-methoxyphenyl)methyl]acetamide
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-propylpiperazine