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1-[2-({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)pyrimidin-4-yl]pyrrolidin-3-ol
N-(butan-2-yl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}-3,4-dihydroquinazolin-4-one
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-{3-[(5-methylpyridin-2-yl)amino]propyl}urea
6-[(1-{[2-(dimethylamino)ethyl](methyl)amino}hex-5-en-2-yl)oxy]-N,N-dimethylpyrazine-2-carboxamide
1-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazol-3-yl]ethan-1-one
4-({1-[(3-acetylphenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
3-(1-butyl-3-methyl-1H-pyrazol-5-yl)-1-[3-(morpholin-4-yl)propyl]urea
2-methyl-5-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-{[4-(4-butyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}piperidine-4-carboxamide
8-chloro-2-(furan-2-yl)-N-(1,2-oxazol-5-ylmethyl)quinoline-4-carboxamide
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-propanoylphenoxy)acetamide
4-(4-chlorophenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]butanamide
3-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propane-1,2-diol
1-[2-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
5-chloro-2-(2-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrrol-1-yl)pyridine
ethyl 1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[1-(2,5-difluorophenyl)cyclopropyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[1'-(2-phenoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
[1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]methanol
6-methoxy-3-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
1-cyclopropanecarbonyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-[(5-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}furan-2-yl)sulfanyl]pyrimidine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
N-benzyl{[2-(1-hydroxyethyl)-1-methyl-1H-1,3-benzodiazol-5-yl]amino}sulfonamide
2-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1-methyl-1H-1,3-benzodiazole
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,2,6-trimethylpyridine-4-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-(4-ethoxyphenyl)ethan-1-one
4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholine
8-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
6-[(3-methoxyphenyl)methoxy]-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-(2-phenylethyl)-1,4-diazepan-2-one
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(morpholin-4-yl)propan-1-one
N-(oxolan-2-ylmethyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)-N-(thiophen-3-ylmethyl)propanamide
1-(4,6-dimethylpyrimidin-2-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidin-4-amine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
methyl 2-[4-(pyrimidin-2-yloxy)phenyl]-1H-1,3-benzodiazole-6-carboxylate
7-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(methylamino)acetamide
(3S,4R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
[(5-ethylpyridin-2-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-4-(pyridin-3-yl)pyrimidine
4-benzyl-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(6,8-dimethoxy-4-methylquinolin-2-yl)-4-(2,2-dimethyloxane-4-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-aminoethyl)-N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H-1,2,3-triazole-4-carboxamide