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3-butanamido-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
2-{4-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[2-methyl-5-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
8-(4-methylpyridine-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]urea
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(1H-pyrazol-3-yl)piperidine
N-(1-hydroxy-2-methylpropan-2-yl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-{1'-[(2-aminopyridin-3-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
1-(3-chlorophenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-ethylpiperazin-2-one
2-(2,3-dihydro-1-benzofuran-5-yl)-N-ethylpyrimidin-4-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1,3-dimethyl-N-(oxan-4-yl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-{1-[(5-chlorofuran-2-yl)methyl]piperidine-3-carbonyl}pyridine
7-(2-benzyl-1,3-thiazole-4-carbonyl)-2-oxa-7-azaspiro[4.5]decane
N-(3-methanesulfonamidophenyl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
3-(3,4-dimethoxyphenyl)-4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrazole
1-[4-({3-[2-(methylsulfanyl)ethyl]-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl}methyl)phenyl]-1H-1,2,3,4-tetrazole
9-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
3-{methyl[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]amino}-1-phenylpropan-1-ol
N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
6-[3-chloro-5-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(3-methoxypropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-amine
1-[1'-(dimethyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-(quinolin-3-yl)urea
N-[2-(piperidin-1-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
(4aS,8aR)-1-(2-aminoethyl)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}oxane-2-carboxamide
9-(2-ethoxypropanoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-1-(1,2,3-thiadiazole-4-carbonyl)piperidine
7-methyl-2-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-2,7-diazaspiro[4.5]decan-6-one
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(2-methoxyphenyl)methyl]urea
6-(methylsulfanyl)-2-(pyrrolidine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2,8-dimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]quinoline-4-carboxamide
2-amino-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-4-phenylpyrimidine-5-carboxamide
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1-phenylpropan-1-one
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
methyl 2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
N-(2-{[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
N-({5-[(1,4-dimethylpiperidin-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide