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1-{3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
[(3S,5R)-1-(4-methoxy-3,5-dimethylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
3-[1-(2-methanesulfonylethyl)-1H-1,2,3-triazol-4-yl]benzonitrile
2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-5-methoxy-4H-pyran-4-one
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-oxo-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-[(3R,4S)-1-(2,5-difluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
9-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-hydroxybenzamide
2-cyclopentyl-9-(3,4-difluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(3-hydroxy-2,2-dimethylpropyl)amino]methyl}piperidin-2-one
3-{[1-(2-methyl-2-phenylpropanoyl)pyrrolidin-3-yl]methyl}benzamide
N-[(3-fluoro-4-methoxyphenyl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-(azocan-1-yl)-3-(2-methoxy-5-{[(1-propylpiperidin-4-yl)amino]methyl}phenoxy)propan-2-ol
1-({[2-(2-ethoxyethoxy)phenyl]carbamoyl}amino)cycloheptane-1-carboxamide
4-ethyl-5-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-2-methyl-1,3-thiazole
methyl 1-(2-methoxyethyl)-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N-cyclopentyl-3-[1-(2-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]propanamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(1-phenylbutyl)benzamide
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](pyridin-2-ylmethyl)amine
3-methyl-6-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridazine
2-[(4-fluorophenyl)methyl]-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}morpholine
N-[(3R,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(propylsulfanyl)acetamide
2-methyl-4-{3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
1,8-bis(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-4-(thiophen-3-yl)phenoxy)acetic acid
1-cyclopentyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
5-({[(2-chloro-3,6-difluorophenyl)methyl](propan-2-yl)amino}methyl)pyrrolidin-2-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[1-(pyridin-2-yl)ethyl]amine
4-{2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}morpholine-2-carboxamide
5-{[4-(2-ethylphenyl)piperazin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
2-[(isoquinolin-5-yloxy)methyl]-N-(1H-1,2,4-triazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-[(4-chlorophenyl)methyl]-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-3-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(4-fluorophenyl)methyl](prop-2-en-1-yl)amine
2-chloro-4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
N-(4-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}phenyl)acetamide
4-(4-methylphenyl)-N-(oxan-4-ylmethyl)-5-(pyridin-4-yl)pyrimidin-2-amine
(1S,5R)-3-[2-(1H-indol-3-yl)ethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
6-{[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]methyl}pyrimidin-4-ol
4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
methyl 1-oxo-2-(pyrimidin-2-ylmethyl)-1,2-dihydroisoquinoline-7-carboxylate
4-{3-[cyclopentyl(prop-2-en-1-yl)amino]propanamido}benzamide
(2S)-3-hydroxy-2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}propanamide
2-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)-6-methylquinolin-4-ol