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N-[(2-fluorophenyl)methyl]-1-methyl-5-(4-methylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(piperidin-3-yl)morpholine
3-[1-(3-fluoropyridine-4-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[2-(dimethylamino)ethyl]-4-(1-methyl-1H-indazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
6-methyl-2-[2-(morpholin-4-ylmethyl)phenoxy]pyridine-3-carbonitrile
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
3-{4-[6-(dimethylamino)pyrimidin-4-yl]piperazin-1-yl}propanamide
4-hydroxy-2-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-5-[3-(dimethylamino)pyrrolidine-1-carbonyl]piperidine-3-carboxamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
2-amino-4-{[(2R)-oxolan-2-ylmethyl]amino}quinazoline-6-carboxylic acid
1-ethyl-4-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}piperidine
2-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
8-(cyclopropylmethyl)-N-(3-methoxyphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-{3-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]piperidin-1-yl}acetamide
ethyl 2-[1-(2,2-dimethylpropyl)-4-(4-fluorobenzenesulfonyl)piperidin-4-yl]acetate
4-(1-methyl-1H-imidazol-5-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(pyridin-3-yl)propyl]benzamide
1-(4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}butan-2-yl)pyrrolidine
(1S,5R)-3-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(benzyloxy)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidine
N-[4-(4-{[2-(1H-imidazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
8-acetyl-2-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(4aS,8aR)-6-[(2,5-difluorophenyl)methyl]-1-propyl-decahydro-1,6-naphthyridin-4a-yl]methanol
1-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
8-[(4-methanesulfonylphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
3-{5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-(cyclohex-1-ene-1-carbonyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
4-methoxy-3-(3-methyl-3-phenylpiperidine-1-carbonyl)benzene-1-sulfonamide
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-[2-(pyridin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3R,4S)-1-(5-fluoro-2-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropyl-N-propylacetamide
5,7-dimethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
N4-[(1-benzylpiperidin-3-yl)methyl]-6-methylpyrimidine-2,4-diamine
2-(2-{[1-(1H-imidazol-1-yl)propan-2-yl]amino}ethyl)-1,2,3,4-tetrahydrophthalazine-1,4-dione
N-(furan-2-ylmethyl)-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyridine-2-carboxamide
6-(3-chlorophenyl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4aR,8aR)-2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[4-({[2-(1H-1,3-benzodiazol-2-yl)ethyl](methyl)carbamoyl}methoxy)phenyl]propanamide
7-(3-methoxypropyl)-2-(6-oxo-1,6-dihydropyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-oxoethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
N,N-dimethyl-4-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]piperazine-1-sulfonamide
(1S,5R)-6-methyl-3-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine