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4-(cyclopropylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-[(2,6-dimethylpyrimidin-4-yl)formamido]-N-(2-methoxyphenyl)propanamide
1-[4-methyl-2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)pyrimidin-5-yl]ethan-1-one
5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}pyrimidin-2-amine
(2E)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyridin-4-yl)prop-2-enamide
N-(2-benzylphenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
1-(methoxymethyl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclobutane-1-carboxamide
methyl(pyridin-3-ylmethyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
7-(1,3-benzothiazol-2-yl)-4-(4-hydroxybutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
(3R)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
9-[2-(morpholin-4-yl)-2-oxoethyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(1-phenylpiperidin-4-yl)piperidin-4-yl]propanamide
7-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
2-[4-(3-methoxypropyl)piperidin-1-yl]-5-methylpyrimidine
N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-7-[(quinolin-5-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
2-{[(1R)-1-(4-methoxyphenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(2S)-2-amino-N-[3-(3,5-dimethylphenoxy)propyl]-3-(1H-imidazol-4-yl)-N-methylpropanamide
methyl 2-[(3-fluoro-4-methylphenyl)sulfamoyl]-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methyl-2-phenylpropan-1-one
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1-cyclopropylethyl)acetamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}methanesulfonamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(2-methanesulfonylethyl)piperazine
9-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-[2-(dimethylamino)ethyl]-N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-oxopyrrolidine-3-carboxamide
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
2-ethyl-9-[2-(2-methoxyphenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(2,4,5-trimethylbenzoyl)-1,4-diazepan-5-one
8-[3-(5-methylfuran-2-yl)butyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpyridine-3-sulfonamide
2-{5-[(2-amino-4-methyl-1,3-thiazol-5-yl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}benzoic acid
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
methyl 2-(1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}-N-methylformamido)acetate
N-{5-[(1E)-pent-1-en-1-yl]pyridin-2-yl}acetamide
3-cyclopropyl-6-[3-(thiophen-2-yl)propyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
8-(2-methyl-1H-pyrrole-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-3-(thiophen-2-yl)-1H-pyrazole
1-(2-methylpyrimidin-4-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
(4aR,7aS)-1-propyl-4-{[4-(pyridin-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-N-[(4-fluorophenyl)methyl]-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-1H-indole-6-carboxamide
3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
1-[2-(pyridin-2-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one