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(1H-imidazol-2-ylmethyl)(methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
1-(3-chlorophenyl)-4-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
2-{[5-(1-methoxyethyl)-4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
(furan-3-ylmethyl)[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
(1S,5R)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2H-1,3-benzodioxol-5-yl)-N-butyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
ethyl 5-[(1,2-oxazol-3-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylate
2-(ethylamino)-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]pyrimidine-5-carboxamide
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
(3S,4S)-1-[(2-methylpyrimidin-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
3-[(5-ethylpyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2,5-dimethylphenyl)ethan-1-one
{2,2-dimethyl-3-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]propyl}dimethylamine
3-{[4-(2,2-dimethylpropanoyl)piperazin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
1-(2-methoxyphenyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-methyl-4-{3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidine
2-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-[4-(3-methylphenyl)piperazin-1-yl]acetamide
N,N-dimethyl-2-[1-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-methoxy-N-(oxolan-2-ylmethyl)propanamide
4-(pyrrolidin-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]butanamide
4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N-methylbutanamide
2-amino-4-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-6-(propan-2-yl)pyridine-3-carbonitrile
4-acetyl-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]benzamide
7-(1-benzothiophen-3-yl)-4-cyclobutanecarbonyl-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2,6-dimethoxy-3-[5-(methoxymethyl)-3-methyl-1H-pyrazol-4-yl]pyridine
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyridine
4-(azocane-1-carbonyl)-1-ethyl-1,2-dihydropyridin-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-ethoxy-4-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}phenol
2-[3-({3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenoxy]acetamide
3-(3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl)-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
5-acetyl-N-[1-(cyclohex-1-en-1-yl)ethyl]thiophene-3-carboxamide
N-cyclopropyl-4-{[4-(pyridin-2-yl)phenyl]methyl}piperazine-2-carboxamide
1-{3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]phenyl}ethan-1-one
4-(2H-1,3-benzodioxol-5-yloxy)-1-(4-methylpyrimidin-2-yl)piperidine-4-carboxylic acid
4-phenyl-5-[3-(1H-pyrazol-3-yl)phenyl]-1H-imidazole
5-(4-chloro-2-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-(4-{2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
9-[(4-ethylphenyl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3,5-dimethylphenyl)-3-{[2-(dimethylsulfamoyl)ethyl]amino}propanamide
4-ethyl-1-methyl-3-[1-(1-methyl-1H-indazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
3-{[(1,3-dihydroxypropan-2-yl)amino]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
1-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}urea