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2-(1H-1,2,3,4-tetrazol-5-yl)-N-(thiolan-3-yl)benzamide
1-[(2-methylphenyl)methyl]-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-(pyridine-2-carbonyl)piperidine-4-carboxamide
1-[1-ethyl-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
N,N,1-trimethyl-6-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-ethyl-N-[2-(2-fluorophenyl)ethyl]-1H-pyrazole-4-carboxamide
1-(2-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-{[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-6-fluorobenzamide
4-(3-hydroxy-3-methylbutyl)-N-(1-methyl-6-oxopiperidin-3-yl)benzamide
methyl 5-{[(3,5-dimethylphenyl)carbamoyl]carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-[(2R,3R,6R)-5-[(2,3-difluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidine-3-carboxamide
1,3,5-trimethyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
(4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)methanol
N-(3,3-diphenylpropyl)-1-ethyl-5-oxopyrrolidine-3-carboxamide
2-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-3,5-difluoropyridine
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(piperidine-1-carbonyl)pyridine
5-[2-(adamantan-1-yl)acetyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-{1-[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(propan-2-ylsulfanyl)acetamido]acetic acid
5-methyl-2-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenol
3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(cyclohexylmethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(2R)-3-methylbutan-2-yl]benzamide
N-(3-ethoxy-2-hydroxypropyl)-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(2,5-dimethylfuran-3-yl)-5-(thiophene-3-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[(5-{1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
4-[2-(benzenesulfonyl)ethyl]-1-[(2,5-dimethylphenyl)methyl]-1,4-diazepan-5-one
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,4-tetrahydroquinolin-2-one
6-[(3R,4S)-3-(2-carboxyethyl)-4-(morpholin-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
1-tert-butyl-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
2-[(4-methoxyphenyl)methyl]-N-(2,2,2-trifluoroethyl)-1,3-benzoxazole-6-carboxamide
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2-diphenylacetamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]morpholine
1-[(2-aminopyridin-3-yl)methyl]-4-(1H-pyrazole-3-carbonyl)-1,4-diazepane-6-carboxylic acid
1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(morpholin-2-yl)ethan-1-one
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]thiophen-3-amine
3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-1-{[3-(pyrrolidin-1-yl)phenyl]methyl}urea
2-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
6-{[(2S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]oxolan-2-yl]methyl}naphthalen-2-ol
5-{1-[(4-chlorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}-4-methylpyrimidin-2-amine
5-(2-chloro-4-methoxyphenoxymethyl)-3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazole
N-(4-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)acetamide
1-(furan-2-ylmethyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}piperidine-3-carboxamide