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4-[({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]benzene-1-sulfonamide
2-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}morpholine
1-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-6-carboxamide
1-(2-phenoxyethyl)-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazole
6,7-dimethyl-2-{[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-1H-1,3-benzodiazole
3-{[1-tert-butyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(2-{2-[5-(2-chlorophenyl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[methyl({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl})amino]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
(4aS,8aR)-1-(carboxymethyl)-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-{1-[1-(naphthalene-2-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
3-(morpholine-4-sulfonyl)-5-(3-phenyl-1H-pyrazol-1-yl)benzoic acid
ethyl 1-(2-methoxyethyl)-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(1H-1,2,3-benzotriazol-4-yl)-4-(6-ethylpyrimidin-4-yl)piperazine-1-carboxamide
5-ethyl-2-methyl-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-4-amine
2-({[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
N-(2-fluorophenyl)-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1-methyl-1H-indol-3-yl)acetamide
3-(2-fluorophenyl)-5-(propan-2-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1,5,6-trimethyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6,8-difluoroquinoline
1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
N-cyclohexyl-3-{[3-(dimethylamino)propyl](methyl)amino}piperidine-1-carboxamide
3,5-dimethyl-1-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,4-triazole
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S)-2-[1-(3-cyclopentaneamido-4-methylphenyl)-N-methylformamido]propanoic acid
1-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-methylpiperazine-2-carboxylic acid
1-cycloheptyl-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
6-(propan-2-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyridazin-3-amine
2-(2,4-difluorophenoxy)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}acetamide
1-(3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}phenyl)ethan-1-one
N-[(3-methoxyphenyl)methyl]-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}propanamide
5-(2-{[4-methyl-4-(methylsulfanyl)pentan-2-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
5-{2-[2-(cyclopentylamino)ethyl]morpholin-4-yl}-2-methyl-2,3-dihydropyridazin-3-one
(4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholin-2-yl)methanamine
1-[2-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
(4aR,7aS)-1-{2-[(cyclohexylmethyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-6-methyl-2-(oxane-4-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N,N-dimethyl-2-{[2-(pyridin-4-ylsulfanyl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
2-{1-[(2-fluorophenyl)methyl]-4-[1-(furan-2-ylmethyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1'-[(2-fluoro-4-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
1-{4-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-(2-methoxyethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-[2-(1H-imidazol-4-yl)ethyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide