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N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-oxoazepan-3-yl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]sulfamoyl}-N,N-dimethylbenzamide
1-methyl-3-(2-methylpropyl)-N-[4-(oxolan-2-yl)butyl]-1H-pyrazole-5-carboxamide
4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
2-(3,4-dichlorophenyl)-4-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-2-methyl-1H-1,3-benzodiazole
[(3R,4R)-1-(4-chloro-3-methylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(2-chlorophenoxy)-1-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
1-(2-methylpropanoyl)-3-(3-phenylpropyl)piperidine-3-carboxylic acid
(1-{1-[4-(5-methylfuran-2-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
N-(2-acetylphenyl)-3-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}propanamide
2-(3-chloro-4-ethoxyphenyl)-1H-1,3-benzodiazole-5-carbonitrile
1-(furan-2-ylmethyl)-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(3R,4S)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzothiazole
2-cyclopropyl-9-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(2-butoxyacetyl)-1-(2-methylphenyl)piperazin-2-one
4-({4-methyl-5-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-cyano-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}benzamide
1-(naphthalen-1-yl)-4-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}butane-1,4-dione
(1R,6S)-6-{[1-(3-phenylphenyl)piperidin-4-yl]amino}cyclohex-3-ene-1-carboxamide
N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-(ethylamino)-N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyrimidine-5-carboxamide
3-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
6-[4-({[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(morpholin-4-yl)butan-1-one
4-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}benzoic acid
4-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)thiomorpholine
1'-[(6-chloro-2H-chromen-3-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-3-[(dimethylcarbamoyl)methyl]-N-(2-ethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
{1-[(4-methoxypiperidin-1-yl)sulfonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
3-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
2-methyl-2-(methylamino)-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}propanamide
methyl 6-(2-fluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 6-[(3-methoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
5-{[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2-[(4-methylphenyl)amino]-4,5-dihydro-1,3-thiazol-4-one
5-methyl-3-[4-({4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]-1,2,4-oxadiazole
N-(2,3-dihydro-1H-inden-2-yl)-4-hydroxy-N-methyl-2-(phenoxymethyl)pyrimidine-5-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(thiophene-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
2-{4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]morpholin-3-yl}acetic acid
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
7-[2-(2H-1,3-benzodioxol-5-yloxy)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]propanoic acid