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1-(2-methylpropyl)-2-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole
(3S,4R)-3-ethyl-4-methyl-1-[2-(pyridin-4-yl)quinoline-4-carbonyl]piperidin-4-ol
1-(furan-2-carbonyl)-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
2-(2-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
7-[(3-methoxyphenyl)methyl]-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[1-(oxan-4-yl)piperidin-3-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N,N-dimethyl-2-{[(oxan-4-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[4-({4-[3-(5-methylfuran-2-yl)butyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
1-(2-methylphenyl)-4-[6-oxo-1-(prop-2-en-1-yl)piperidine-3-carbonyl]piperazin-2-one
2-(4-hydroxyphenyl)-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
3-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
7-methyl-2-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
9-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
2-benzyl-8-(2-propoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1R,2S)-2-phenylcyclohexyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-ethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrimidine-5-carboxamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]methanol
1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
1-[(3-methoxyphenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
5-(8-methoxy-2H-chromen-3-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-{2-[(4-methyl-1,4-diazepan-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-(4-methylphenyl)-4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-2-one
2-(4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)acetamide
2-{[1-(4-oxo-3,4-dihydroquinazolin-3-yl)propan-2-yl]amino}-N-(propan-2-yl)acetamide
N-methyl-1,1-dioxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1λ6-thiane-4-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(1H-imidazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
(2S,4R)-4-amino-N,N-diethyl-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidine-2-carboxamide
1-[3-(1H-imidazol-1-yl)propyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(1-hydroxycyclohexyl)methyl]piperidine-4-carboxamide
(1S,3R)-3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]cyclohexan-1-amine
1-[2-(1H-imidazol-2-yl)benzoyl]-4-[2-(methylsulfanyl)ethyl]piperazine
2-{2-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrrol-1-yl}-1,3-thiazole
6-{[3-(1H-1,2,4-triazol-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-methoxy-1,3-benzothiazol-2-amine
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-ethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]acetamide
3-chloro-2-[3-(propan-2-yloxy)phenyl]pyridine
1-benzoyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]piperidin-4-amine
N-methyl-2-propyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3-thiazole-4-carboxamide
4-benzyl-3-ethyl-1-(2-propylpyridine-4-carbonyl)-1,4-diazepan-5-one
4-(2,6-dimethylpyridin-3-yl)-N-[(1R,2S)-2-phenylcyclopropyl]pyrimidin-2-amine
8-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-[8-(1-benzothiophen-2-ylmethyl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
(2S,4S)-4-amino-N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methylpyrrolidine-2-carboxamide
ethyl 4-({4-[2-(2-fluorophenyl)ethyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}amino)piperidine-1-carboxylate