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dimethyl({2-[2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl})amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
2-(methylamino)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyridine-4-carboxamide
1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(quinazolin-4-yloxy)ethan-1-one
N-[(3R,4R)-1-[(2-aminopyridin-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-[2-(2-fluorophenoxy)ethyl]-3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
3-{2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
(2E)-3-(3,4-dimethoxyphenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]prop-2-enamide
N-[3-(1H-indazol-1-yl)propyl]-1,7-dimethyl-1H-indole-2-carboxamide
1-[1-(2-phenylpropyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(3-{3-[1-(dimethylamino)ethyl]phenyl}thiophen-2-yl)ethan-1-one
3-[(2-fluorophenyl)formamido]-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-(thiophen-3-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(2S,4S)-4-amino-N-methyl-1-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}pyrrolidine-2-carboxamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidine
1-(3,3-diphenylpropyl)-5-{2-[(pyridin-2-ylmethyl)amino]ethyl}pyrrolidin-2-one
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6,8-dimethylquinoline
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
(4aS,8aR)-6-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
5-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-cyclopropyl-N-[2-(2-ethoxyphenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
3-[3-(1H-imidazol-1-yl)propyl]-1-(3-methanesulfonamido-4-methoxyphenyl)urea
2-(benzyloxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-methyl-4-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]piperazine
2-(dimethylamino)-2-(2-methylphenyl)-1-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
3-hydroxy-1-(2-methoxyethyl)-3-({3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)piperidin-2-one
(3S,4R)-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[2-({2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}amino)ethyl]pyridine-3-carboxamide
3-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-4-methoxy-N-methylbenzamide
11-methyl-4-(2-oxooxolan-3-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
N-(oxolan-3-ylmethyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-8-fluoroquinoline-2-carboxamide
1-oxo-2-[2-(piperidin-1-yl)ethyl]-N-[(3R)-pyrrolidin-3-yl]-2,3-dihydro-1H-isoindole-5-carboxamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-sulfonyl]-2,1,3-benzothiadiazole
2-(naphthalen-2-yloxy)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}propanamide
1-(2-ethoxyphenyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
(3S,4S)-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4-(naphthalen-2-yl)piperidin-3-ol
N-(2-methoxyethyl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(propan-2-yl)piperidine-3-carboxamide
{4-[2-(benzyloxy)phenyl]pyridin-2-yl}methanol
(3R,4S)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-cyclopropylpyrrolidin-3-amine
2-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide