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1-methyl-6-(pyridin-4-yl)-N-[1-(thiophen-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,5R,9R)-5-hydroxy-11-(3-methoxybenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
[(4-fluoro-3-methylphenyl)methyl](methyl)[1-(pyridin-2-yl)propyl]amine
5-fluoro-N,N-dimethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
4-(4-fluorophenyl)-2-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-1,3-thiazole
3-(4-fluorophenyl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
3-(2-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
(2S,4R)-4-(dimethylamino)-1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]pyrrolidine-2-carboxylic acid
2-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
2-(3-methyl-1,2-oxazol-5-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
(2S)-4-(methylsulfanyl)-2-{[2-(phenylamino)pyrimidin-5-yl]formamido}butanoic acid
5-(3-fluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
2-{[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}benzoic acid
N-methyl-N-[1-(pyridin-2-yl)propyl]-2,1-benzoxazole-3-carboxamide
2-{3-[3-(6-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(1,3-thiazol-2-yl)propanamide
2-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-3-ol
4,6-dimethyl-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
1-[3-({3-[2-(2-methoxyethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
4,5-dimethyl-6-[3-(pyridin-3-yl)azetidin-1-yl]-2-(pyrrolidin-1-yl)pyrimidine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-hydroxyethyl)piperidine-4-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-chloro-N-(2-methoxyethyl)benzamide
N-methyl-4-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)benzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(prop-2-en-1-yl)acetamide
1-cyclopentyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-6-oxopiperidine-3-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(3-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(3-methoxypropyl)-9-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-4-methyl-1,4-diazepane
2-acetyl-8-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(4-fluoro-3-methylphenyl)-5-(methanesulfonylmethyl)pyridine
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]-1-(3-phenylpropyl)piperidin-2-one
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
N-(2,4-dimethoxyphenyl)-6-oxopiperazine-2-carboxamide
2-({3-[(6,8-dimethoxy-4-methylquinolin-2-yl)amino]propyl}(2-hydroxyethyl)amino)ethan-1-ol
2-amino-8-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[2-(1H-imidazol-4-yl)ethyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(furan-2-ylmethyl)acetamide
3-{1-[1-(carbamoylmethyl)piperidin-4-yl]-N-methylformamido}-3-phenylpropanoic acid
5-{2-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(2-fluorophenyl)methyl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methoxy-1-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-1,2-dihydropyridin-2-one
4-[2-(2,5-dimethoxyphenyl)ethyl]thiomorpholine
N-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
(3R,4S)-4-[methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})amino]oxolan-3-ol