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6-methyl-2-oxo-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridine-3-carbonitrile
5-methanesulfonyl-2-methyl-4-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidine
3-(3-methoxyphenyl)-5-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazole
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(4-phenylphenyl)acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}pyrrolidin-3-yl]acetamide
1-(azocan-1-yl)-3-[5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
4-[3-(2-methoxyphenoxy)propyl]-1-(3-methoxyphenyl)piperazin-2-one
6-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-{[cyclohexyl(thiophen-2-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
N-[(3S,4R)-1-(1-acetylpiperidine-4-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(3S,4R)-4-(2-methoxyphenyl)-1-(5-methyl-1-benzofuran-2-carbonyl)pyrrolidine-3-carboxylic acid
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[(3,5-dimethylphenyl)methyl]-4-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperazin-2-one
[(1S)-1-[1-(3-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl](methyl)amine
3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
1-{2-[(5-fluoroquinazolin-4-yl)amino]ethyl}imidazolidin-2-one
(2R,3R)-3-amino-1'-[(5-ethylpyridin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-propyl-1,3,4-oxadiazol-2-amine
[(2,3-dimethyl-1H-indol-7-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(1,2-oxazolidin-2-yl)pyridine
2-(azocan-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
8-[(2R)-2-hydroxypropanoyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-chloro-4-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(oxan-4-yl)piperazine
(3S,4R)-1-[(3-chloro-4-methoxyphenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
3-(1-{imidazo[1,2-a]pyridin-3-ylmethyl}-4-phenyl-1H-imidazol-5-yl)benzonitrile
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-{4-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-ethyl-N-methylpyrimidine-5-carboxamide
1-ethyl-8-[(4-hydroxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-{4-[(5-methylfuran-2-yl)methyl]morpholin-3-yl}acetamide
2-(4-fluorophenyl)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]azetidine
2-[2-chloro-4-(2-methoxypyridin-3-yl)phenoxy]propanoic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-methoxy-4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridine
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-5-propyl-1,2-oxazole-4-carboxamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
1-(2-oxo-2-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
(2R)-2-amino-3-hydroxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
methyl 1-methyl-4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-pyrazole-5-carboxylate
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
5-cyclopropyl-N,N-diethyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
1-(cyclohexylmethyl)-4-[(oxan-4-yl)amino]pyrrolidin-2-one
(2S)-2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-(2,2-diphenylethyl)-4-(2-methoxyethyl)-1,4-diazepan-5-one
4-{2-[(E)-2-phenylethenyl]pyridine-4-carbonyl}morpholine