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1-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2,6-dimethylpyridin-4-yl)piperazine
4-[3-(benzyloxy)azetidine-1-carbonyl]-1-tert-butylpyrrolidin-2-one
N-(1-{1-[(2S)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-phenylmethanesulfonamide
3-ethyl-1-(4-fluorophenyl)-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-cyclopropyl-1-(2-{1-[3-(3,4-dimethoxyphenyl)propanoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-{1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
3-(methylsulfanyl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
4-methyl-6-(4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-1-yl)pyrimidin-2-amine
methyl 3-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]propanoate
4-(5-methylpyridin-2-yl)-1-(oxolane-3-carbonyl)piperidin-4-ol
methyl 1-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)cyclopropane-1-carboxylate
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(4-chlorophenyl)-4-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-{1-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)ethan-1-one
1-[1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)piperidin-4-yl]pyrrolidin-2-one
N-cyclopropyl-4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
5-(2,4-dimethoxyphenyl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-[(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-{3-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indole
3-hydroxy-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}pyridine-2-carboxamide
4-cyano-1-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrrole-2-carboxamide
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(4-methylpiperazin-1-yl)ethan-1-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(2-methylpropyl)(pyridin-2-ylmethyl)amine
4-[(5-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}ethan-1-ol
2-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)benzoic acid
4-{1-[2-(ethylsulfanyl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,4-dimethyl-5-sulfamoylbenzamide
1-methyl-3-(2-methylpropyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1H-pyrazole-5-carboxamide
2-(4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
N-[1-(2-chlorophenyl)ethyl]-9H-purin-6-amine
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyrazin-2-ol
1-(azepan-1-yl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propan-1-one
5-acetyl-3-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-methylpiperidin-3-ol
1-(2-methoxyethyl)-6-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}piperidine-3-carboxamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
(2R)-2-cyclohexyl-1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-hydroxyethan-1-one
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N,N-diethylpiperidine-3-carboxamide
3-[5-(3-cyclohexylpropanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-(4-methyl-3-phenylpiperazin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(2-methoxyphenyl)propan-1-one
8-methoxy-N-methyl-N-(quinolin-8-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
4-{3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-pyrazole
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyridine-3-carboxamide