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5-{1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-5-methoxyphenol
methyl 4-{[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}benzoate
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidine-2-carboxylate
6-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1,4-diazepane
1-[3-(1H-pyrazol-1-yl)phenyl]-N-[3-(pyridin-2-yl)propyl]piperidin-4-amine
5-(2,4,5-trimethoxybenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
1-[1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-3-yl]-2-phenylethan-1-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
2-[(4aR,7aS)-4-(cyclopropanesulfonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N,N-dimethyl-2-{[3-(methylsulfanyl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[4-(propylsulfamoyl)phenyl]urea
9-[3-(1H-imidazol-1-yl)butanoyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(4-fluoro-3-methylphenyl)-3-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]propanamide
3-(furan-2-ylmethyl)-1-(3-methanesulfonamidophenyl)-3-(2-methylpropyl)urea
3-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}phenol
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(2-methoxyethyl)-3-(1,3-thiazol-2-ylmethyl)urea
1-{4-[3-({[(4-phenylphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
(3aS,6aS)-5-(5-chloro-3-fluoropyridin-2-yl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(3S)-2-oxoazepan-3-yl]amino}-N,N-bis(prop-2-en-1-yl)acetamide
N-[(5-methylfuran-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-3,4-dihydroquinazolin-4-one
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
8-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-ethyl-4-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(4aS,8aS)-2-(isoquinolin-1-yl)-decahydro-2,7-naphthyridin-4a-ol
2-(azepan-1-yl)-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
4-(naphthalen-1-ylmethyl)-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one
methyl N-{1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl}carbamate
(1R,3S)-3-methoxy-7-[4-methyl-6-(methylamino)pyrimidin-2-yl]-7-azaspiro[3.5]nonan-1-ol
N-tert-butyl-5-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
8-chloro-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-2-carboxamide
methyl[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl](oxan-2-ylmethyl)amine
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(2S,4S)-1-(1-benzofuran-2-ylmethyl)-N-ethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[(2R,4R,6S)-2-tert-butyl-6-(2-methoxypyrimidin-5-yl)oxan-4-yl]acetamide
2-amino-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(4-fluorophenyl)methyl]piperidin-4-ol
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
7-(5-chloropyridin-2-yl)-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-amino-4-(1-phenyl-1H-pyrazol-5-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-(1-methylpiperidin-4-yl)piperidine
4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-hydroxypiperidine-4-carboxylic acid
N-cyclopentyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
N-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide