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2-chloro-3-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
(3S,4S)-4-cyclopropyl-1-{2-[4-(trifluoromethyl)phenyl]acetyl}pyrrolidine-3-carboxylic acid
8-[2-(quinazolin-4-yloxy)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-ethyl-5-methyl-N4-[(5-methyl-1H-imidazol-4-yl)methyl]pyrimidine-2,4-diamine
(2S,4R)-N-ethyl-1-[(3-methoxyphenyl)methyl]-4-(3-methyloxetane-3-amido)pyrrolidine-2-carboxamide
9-{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(1R,5R)-6-(1H-1,2,3-benzotriazole-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
8-(1,4-dioxan-2-ylmethyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(oxan-4-yl)-4-[(5-propylfuran-2-yl)methyl]piperazine
4-{1-[2-(1-hydroxyethyl)-1-methyl-1H-1,3-benzodiazol-5-yl]-1H-imidazol-2-yl}-2,6-dimethylphenol
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(3-methylphenyl)methyl]urea
2-(2-pentylpyrimidin-4-yl)pyridine-4-carboxylic acid
N-(propan-2-yl)-3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propanamide
2-[3-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)phenoxy]ethan-1-ol
1-(cyclopropylmethyl)-4-[(4-methoxypyridin-2-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
4-[(1S,2S)-2-hydroxycyclohexyl]-N-[3-(2-methoxyethoxy)phenyl]piperazine-1-carboxamide
1-methyl-5-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
8-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-[ethyl({[4-(2-fluorophenyl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(pyridin-3-yl)acetamide
1-(2-ethylbenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1H-1,3-benzodiazole
2-amino-6-(2-fluoro-4-methoxyphenyl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
3-tert-butyl-4-(6-methoxypyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
N3-(adamantan-2-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclohexyl-3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propanamide
2-(3-hydroxypropyl)-9-(pyrimidin-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-chloro-3-(1-hydroxy-3-methylbutan-2-yl)-3,4-dihydroquinazolin-4-one
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,6-dimethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
6-{[(3R,4S)-4-cyclopropyl-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
1-cyclopentyl-4-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-1,2-oxazolidin-4-ol
3-{[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]amino}-N,N-dimethylazepane-1-carboxamide
3-(3,5-dimethoxyphenyl)-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(methylsulfanyl)pyrimidine
4-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]morpholine
3-(2,3-dimethoxy-5-methylphenyl)-6-(propan-2-yloxy)pyridazine
4-({5-[5-(oxolan-2-yl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
4-{[1-(4-methyl-1,3-thiazol-2-yl)ethyl]sulfamoyl}-N-(propan-2-yl)benzamide
(3S,9aR)-3-(2-methylpropyl)-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione