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5-(4-aminopiperidine-1-carbonyl)-3-methyl-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-(3-chlorophenyl)-N-(1,2-oxazol-5-ylmethyl)-3-phenylpropanamide
N-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]acetamide
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(1-methylpiperidin-3-yl)propanamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
1-(4-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
2-(adamantan-1-yl)-4-hydroxy-N-[3-(methylsulfanyl)propyl]pyrimidine-5-carboxamide
4-[1-(1-carboxycyclopropanecarbonyl)piperidin-3-yl]benzoic acid
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-N,N-dimethyl-2,3-dihydro-1H-inden-2-amine
ethyl 5-({5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}methyl)furan-2-carboxylate
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(3aS,6aS)-2-cyclohexyl-5-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-amino-1-[3-(benzylsulfanyl)propanoyl]-N-methylpyrrolidine-2-carboxamide
(1R,5R)-6-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-(pyrrolidine-1-carbonyl)piperidine
N-[3-(1H-imidazol-1-yl)propyl]-2,6-dimethyl-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
N-[3-(dimethylamino)propyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(furan-3-ylmethyl)-4-(2-phenylpropyl)-1H-1,2,3-triazole
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-(thiolan-3-yl)piperidin-4-amine
3-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]naphthalen-2-ol
7-(2,1,3-benzothiadiazole-4-sulfonyl)-2-oxa-7-azaspiro[4.5]decane
N-tert-butyl-4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}morpholine
1-benzyl-N-(2-fluoroethyl)-4-phenylpiperidine-4-carboxamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}quinoline-3-carboxamide
4-[(2,5-difluorophenyl)methyl]-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3-{[2-(3-methoxyphenyl)ethyl]carbamoyl}phenyl)amino]acetic acid
3-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
4-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(2,5-dimethylphenyl)-1H-imidazol-1-yl]-3-(furan-2-yl)propanoic acid
4-[(2-fluorophenyl)methyl]-1-(1-phenyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
{1-[2-(5-butyl-4-phenyl-1H-imidazol-1-yl)ethyl]piperidin-3-yl}methanol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
4-(cyclohexylmethyl)-3-[hydroxy(phenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
4-(3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-6-phenylpyridin-2-yl)morpholine
4-[6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1-phenylpiperazin-2-one
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-3-(3-methoxyphenyl)-1H-pyrazole
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-{[(1s,4s)-4-aminocyclohexyl]amino}pyridine-3-carboxamide
ethyl 1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(4-hydroxyphenyl)methyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(4-ethylphenyl)propanamide
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
(2S,4S)-N-ethyl-4-[2-(4-hydroxyphenyl)acetamido]-1-[2-(methylsulfanyl)acetyl]pyrrolidine-2-carboxamide
(1S,5R)-3-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1H-1,3-benzodiazol-2-ylmethyl)(2-methoxyethyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]propan-1-one
2-{[5-(2-ethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-6-methyl-3,4-dihydropyrimidin-4-one
1-(4-chlorophenyl)-5-methyl-4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperazin-2-one