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(2-{[4-(1H-indol-4-ylmethyl)piperazin-1-yl]methyl}phenyl)methanol
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-{imidazo[1,2-a]pyridin-2-yl}-N-methylpropanamide
4-methyl-3-{2-[4-(4-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-methylpyridine-3-carboxylic acid
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-5H-chromeno[4,3-b]pyridine-3-carbonitrile
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethylthiophene-2-carboxamide
2,7,8-trimethyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]quinoline-4-carboxamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
6-({[3-(2-amino-1,3-thiazol-4-yl)propyl]amino}methyl)-1,4-oxazepan-6-ol
2-methyl-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)propanamide
4-[3-oxo-3-(pyrrolidin-1-yl)propyl]-N-(quinolin-7-yl)piperidine-1-carboxamide
1-(2-aminoethyl)-N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-methyl-4-[4-(4-phenyl-1H-imidazol-5-yl)phenyl]but-3-yn-2-ol
7-(3-chlorophenyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
methyl[1-(pyrazin-2-yl)propan-2-yl]{[4-(trifluoromethoxy)phenyl]methyl}amine
2-{[propyl(pyridin-3-ylmethyl)amino]methyl}benzonitrile
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[2-(oxan-4-yl)ethyl]acetamide
1-(3-chloro-5-fluorobenzoyl)-3-(2,5-dimethoxyphenyl)pyrrolidine
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](propyl)(pyridin-3-ylmethyl)amine
N,N-dimethyl-6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazin-2-amine
4-[3-carboxy-5-(cyclobutylmethoxy)benzoyl]piperazine-2-carboxylic acid
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
5-(azepane-1-carbonyl)-1-benzyl-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-ethyl-4-[2-oxo-2-(piperidin-1-yl)ethoxy]-N-(pyridin-2-ylmethyl)benzamide
methyl 2-(2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(2-methyl-1H-imidazol-4-yl)methyl](2-methylpropyl)amine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methoxyethan-1-one
2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}acetamide
N-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)acetamide
4-[(4-methanesulfonylphenyl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
4-[1-(1-benzofuran-2-ylmethyl)azetidin-3-yl]pyridine
(2S,4R)-4-(dimethylamino)-N-(2-ethoxyphenyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N'-(2,5-dimethylphenyl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanediamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(methylamino)-N-[2-(naphthalen-1-yl)propan-2-yl]acetamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
2-methyl-N-[3-(morpholin-4-yl)propyl]-2-(thiophen-2-ylformamido)propanamide
8-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-hydroxypropyl)-9-(5-methoxypyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
4-[(4-{[(4-methylphenyl)methyl]amino}quinazolin-2-yl)methyl]piperazine-1-carbaldehyde
1-(3-{[3-(3-hydroxyazetidine-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
2-cyclopropyl-4-methyl-5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}pyrimidine
1-[(3S,4S)-3-hydroxy-4-[(1H-imidazol-2-ylmethyl)(methyl)amino]pyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
8-methoxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(4-methoxyphenyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]cyclopentane-1-carboxamide